TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Kakatiya University
Curated by ChEMBL
Kakatiya University
Curated by ChEMBL
Affinity DataKi: 660nMAssay Description:Inhibition of human MRP1 expressed in Spodoptera frugiperda Sf9 cells assessed as inhibition of NEM-GS-induced vanadate-sensitive ATPase activity mea...More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Kakatiya University
Curated by ChEMBL
Kakatiya University
Curated by ChEMBL
Affinity DataKi: 950nMAssay Description:Inhibition of human MRP1 expressed in Spodoptera frugiperda Sf9 cells assessed as inhibition of NEM-GS-induced vanadate-sensitive ATPase activity mea...More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Kakatiya University
Curated by ChEMBL
Kakatiya University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human MRP1 expressed in Spodoptera frugiperda Sf9 cells assessed as inhibition of NEM-GS-induced vanadate-sensitive ATPase activity mea...More data for this Ligand-Target Pair