Compile Data Set for Download or QSAR
maximum 50k data
Found 33 Enz. Inhib. hit(s) with all data for entry = 50033424
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345056(2-(6-(3-((dimethylamino)methyl)phenyl)-2-(4-fluoro...)
Affinity DataIC50:  1nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345045(CHEMBL1778950 | N-isopropyl-2-(2-(3-methoxyphenyl)...)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345055(2-(6-(5-((dimethylamino)methyl)-2-fluorophenyl)-2-...)
Affinity DataIC50:  7nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345043(2-(6-(3-((dimethylamino)methyl)phenyl)-2-(3-methox...)
Affinity DataIC50:  9nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345048(2-(2-(3-chlorophenyl)-4-oxo-6-(3-(piperidin-1-ylme...)
Affinity DataIC50:  9nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345046(2-(2-(3-chlorophenyl)-6-(3-((dimethylamino)methyl)...)
Affinity DataIC50:  19nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345052(2-(6-(6-((dimethylamino)methyl)pyridin-2-yl)-2-(3-...)
Affinity DataIC50:  37nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345044(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-2-(3-methoxyp...)
Affinity DataIC50:  46nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345050(2-(6-(4-((dimethylamino)methyl)pyridin-2-yl)-2-(3-...)
Affinity DataIC50:  52nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345060(CHEMBL1777825 | N-(cyclopropylmethyl)-2-(4-oxo-2-p...)
Affinity DataIC50:  60nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345047(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-2-(3-chloroph...)
Affinity DataIC50:  60nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345051(2-(6-(5-((dimethylamino)methyl)pyridin-3-yl)-2-(3-...)
Affinity DataIC50:  77nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345059(CHEMBL1778932 | N-(cyclopropylmethyl)-2-(6-(3-(mor...)
Affinity DataIC50:  79nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345040(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-4-oxo-2-pheny...)
Affinity DataIC50:  187nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345042(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-4-oxo-2-pheny...)
Affinity DataIC50:  238nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345034(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-4-oxo-2-pheny...)
Affinity DataIC50:  275nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345032(CHEMBL1778937 | N-(cyclopropylmethyl)-2-(6-(3-((di...)
Affinity DataIC50:  314nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345064(CHEMBL1778936 | N-(cyclopropylmethyl)-2-(6-(3-((me...)
Affinity DataIC50:  320nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345035(CHEMBL1778940 | N-(cyclopropylmethyl)-2-(4-oxo-2-p...)
Affinity DataIC50:  388nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345039(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-4-oxo-2-pheny...)
Affinity DataIC50:  397nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345054(2-(6-(5-((dimethylamino)methyl)thiophen-2-yl)-2-(3...)
Affinity DataIC50:  500nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345033(CHEMBL1778938 | N-(cyclopropylmethyl)-2-(6-(3-((di...)
Affinity DataIC50:  540nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345049(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-2-(2-methoxyp...)
Affinity DataIC50:  610nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345036(CHEMBL1778941 | N-(cyclopropylmethyl)-2-(6-(3-((2-...)
Affinity DataIC50:  642nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345053(2-(6-(5-((dimethylamino)methyl)furan-2-yl)-2-(3-me...)
Affinity DataIC50:  700nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345038(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-4-oxo-2-pheny...)
Affinity DataIC50:  1.04E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345063(2-(6-(3-(aminomethyl)phenyl)-4-oxo-2-phenylquinazo...)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345037(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-4-oxo-2-pheny...)
Affinity DataIC50:  2.35E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345041(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-4-oxo-2-pheny...)
Affinity DataIC50:  2.55E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345057(CHEMBL1778827 | N-(cyclopropylmethyl)-2-(6-(2-(mor...)
Affinity DataIC50: >2.00E+4nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345061(CHEMBL1778933 | N-(cyclopropylmethyl)-2-(6-(4-(mor...)
Affinity DataIC50: >2.00E+4nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345062(CHEMBL1778934 | N-(cyclopropylmethyl)-2-(4-oxo-2-p...)
Affinity DataIC50: >2.00E+4nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50345058(CHEMBL1778828 | N-(cyclopropylmethyl)-2-(4-oxo-2-p...)
Affinity DataIC50: >2.00E+4nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed