Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50033586
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347722BDBM50347722(CHEMBL1802517)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50322727BDBM50322727(4-[(4-{[3-(4-Fluorobenzyl)-2,4-dioxo-1,3-thiazolan...)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347723BDBM50347723(CHEMBL1802518)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347724BDBM50347724(CHEMBL1802519)
Affinity DataIC50: 7.30nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347716BDBM50347716(CHEMBL1802471)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347715BDBM50347715(CHEMBL1802470)
Affinity DataIC50: 10nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347718BDBM50347718(CHEMBL1802473)
Affinity DataIC50: 25nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347721BDBM50347721(CHEMBL1802516)
Affinity DataIC50: 26nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347725BDBM50347725(CHEMBL1802520 | CHEMBL1802521)
Affinity DataIC50: 55nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347725BDBM50347725(CHEMBL1802520 | CHEMBL1802521)
Affinity DataIC50: 59nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347714BDBM50347714(CHEMBL1802469)
Affinity DataIC50: 71nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347713BDBM50347713(CHEMBL1802468)
Affinity DataIC50: 147nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347720BDBM50347720(CHEMBL1802475)
Affinity DataIC50: 683nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347719BDBM50347719(CHEMBL1802474)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAutotaxin(Human)
The Netherlands Cancer Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347717BDBM50347717(CHEMBL1802472)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed