Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50033592
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50418829(CHEMBL1802381)
Affinity DataIC50: 10nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347865(CHEMBL1802383)
Affinity DataIC50: 20nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347864(CHEMBL1802382)
Affinity DataIC50: 60nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347868(CHEMBL1802387)
Affinity DataIC50: 90nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347866(CHEMBL1802384)
Affinity DataIC50: 130nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347870(CHEMBL1802869)
Affinity DataIC50: 390nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347869(CHEMBL1802388)
Affinity DataIC50: 620nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347863(CHEMBL1802870)
Affinity DataIC50: 770nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347868(CHEMBL1802387)
Affinity DataIC50: 920nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347863(CHEMBL1802870)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of hemagglutinin epitope-tagged human Nek2 transfected tetracycline-induced in human HEK293 cells pre-incubated for 45 mins by immunopreci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347866(CHEMBL1802384)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347860(CHEMBL1802386)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347867(CHEMBL1802385)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human Cdk2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347863(CHEMBL1802870)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347861(CHEMBL1802871)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347867(CHEMBL1802385)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347861(CHEMBL1802871)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347862(CHEMBL1802872)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347862(CHEMBL1802872)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347863(CHEMBL1802870)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human Plk1 using dephosphorylated alpha-casein as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50347860(CHEMBL1802386)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed