Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50039478
TargetAurora kinase A(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50353271(CHEMBL1830670)
Affinity DataIC50: 25nMAssay Description:Inhibition of GST-tagged Aurora A kinase expressed in insect cells assessed as inhibition of [33P]gamma-ATP incorporation in substrate after 60 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50353272(CHEMBL1830673)
Affinity DataIC50: 39nMAssay Description:Inhibition of GST-tagged Aurora A kinase expressed in insect cells assessed as inhibition of [33P]gamma-ATP incorporation in substrate after 60 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM22984(Adriamycin | (8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5...)
Affinity DataIC50: 40nMAssay Description:Inhibition of GST-tagged Aurora A kinase expressed in insect cells assessed as inhibition of [33P]gamma-ATP incorporation in substrate after 60 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50353273(CHEMBL1830669)
Affinity DataIC50: 51nMAssay Description:Inhibition of GST-tagged Aurora A kinase expressed in insect cells assessed as inhibition of [33P]gamma-ATP incorporation in substrate after 60 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50353274(CHEMBL1830668)
Affinity DataIC50: 101nMAssay Description:Inhibition of GST-tagged Aurora A kinase expressed in insect cells assessed as inhibition of [33P]gamma-ATP incorporation in substrate after 60 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50353275(CHEMBL1830680)
Affinity DataIC50: 104nMAssay Description:Inhibition of GST-tagged Aurora A kinase expressed in insect cells assessed as inhibition of [33P]gamma-ATP incorporation in substrate after 60 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50353276(CHEMBL1830671)
Affinity DataIC50: 120nMAssay Description:Inhibition of GST-tagged Aurora A kinase expressed in insect cells assessed as inhibition of [33P]gamma-ATP incorporation in substrate after 60 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Umm Al-Qura University

Curated by ChEMBL
LigandPNGBDBM50353277(CHEMBL1830681)
Affinity DataIC50: 9.24E+3nMAssay Description:Inhibition of GST-tagged Aurora A kinase expressed in insect cells assessed as inhibition of [33P]gamma-ATP incorporation in substrate after 60 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed