Compile Data Set for Download or QSAR
Report error Found 295 Enz. Inhib. hit(s) with all data for entry = 50033763
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350866(CHEMBL1819441)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350852(CHEMBL1817706)
Affinity DataEC50:  0.105nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350876(CHEMBL1819542)
Affinity DataEC50:  0.123nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350869(CHEMBL1817704)
Affinity DataEC50:  0.126nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350874(CHEMBL1819540)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350866(CHEMBL1819441)
Affinity DataEC50:  0.155nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350853(CHEMBL1817707)
Affinity DataEC50:  0.162nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350852(CHEMBL1817706)
Affinity DataEC50:  0.210nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350875(CHEMBL1819541)
Affinity DataEC50:  0.234nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350868(CHEMBL1819555)
Affinity DataEC50:  0.25nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350851(CHEMBL1817705)
Affinity DataEC50:  0.260nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350876(CHEMBL1819542)
Affinity DataEC50:  0.270nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350851(CHEMBL1817705)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350872(CHEMBL1817761)
Affinity DataEC50:  0.320nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350849(CHEMBL1817702)
Affinity DataEC50:  0.340nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350865(CHEMBL1819440)
Affinity DataEC50:  0.350nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350869(CHEMBL1817704)
Affinity DataEC50:  0.380nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350865(CHEMBL1819440)
Affinity DataEC50:  0.450nMAssay Description:Agonist activity at recombinant human vasopressin V2 receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350877(CHEMBL1819543)
Affinity DataEC50:  0.490nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350882(CHEMBL1819548)
Affinity DataEC50:  0.540nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350864(CHEMBL1819439)
Affinity DataEC50:  0.540nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350870(CHEMBL1817709)
Affinity DataEC50:  0.550nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350853(CHEMBL1817707)
Affinity DataEC50:  0.570nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350906(CHEMBL1819549)
Affinity DataEC50:  0.617nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350871(CHEMBL1817756)
Affinity DataEC50:  0.620nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350872(CHEMBL1817761)
Affinity DataEC50:  0.690nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350865(CHEMBL1819440)
Affinity DataEC50:  0.690nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350867(CHEMBL1819554)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350854(CHEMBL1817708)
Affinity DataEC50:  0.820nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350849(CHEMBL1817702)
Affinity DataEC50:  0.891nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350887(CHEMBL1819556)
Affinity DataEC50:  0.940nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350861(CHEMBL1817754)
Affinity DataEC50:  1nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350842(CHEMBL1817695)
Affinity DataEC50:  1nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350891(CHEMBL1819560)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350859(CHEMBL1817752)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350873(CHEMBL1817770)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350866(CHEMBL1819441)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at recombinant human vasopressin V2 receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350862(CHEMBL1817755)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350839(CHEMBL1817692)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350905(CHEMBL1817772)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350842(CHEMBL1817695)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350856(CHEMBL1817749)
Affinity DataEC50:  2nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350868(CHEMBL1819555)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350845(CHEMBL1817698)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350883(CHEMBL1819550)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350870(CHEMBL1817709)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at human OT receptor expressed in CHO-K1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350860(CHEMBL1817753)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350870(CHEMBL1817709)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350871(CHEMBL1817756)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50350858(CHEMBL1817751)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
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