Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50033717
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419019BDBM50419019(CHEMBL1814294)
Affinity DataEC50:  2.00E+3nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350149BDBM50350149(CHEMBL1814312)
Affinity DataEC50:  3.80E+3nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419030BDBM50419030(CHEMBL1814310)
Affinity DataEC50:  7.70E+3nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81558BDBM81558(Magreth-11a)
Affinity DataEC50:  8.40E+3nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350150BDBM50350150(CHEMBL1814307)
Affinity DataEC50:  9.20E+3nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419021BDBM50419021(CHEMBL1814308)
Affinity DataEC50:  9.30E+3nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419022BDBM50419022(CHEMBL1814306)
Affinity DataEC50:  1.24E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50295920BDBM50295920(CHEMBL555297 | Magreth-1 | 4'-Methoxy-5,3'-dipropy...)
Affinity DataEC50:  1.27E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81563BDBM81563(Magreth-16a)
Affinity DataEC50:  1.43E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81565BDBM81565(Magreth-17a)
Affinity DataEC50:  1.48E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81559BDBM81559(Magreth-11b)
Affinity DataEC50:  1.69E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419020BDBM50419020(CHEMBL1814309)
Affinity DataEC50:  1.85E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50295924BDBM50295924(4'-Methoxy-3'-(Z)-propenyl)-5-(2-propenyl)-bipheny...)
Affinity DataEC50:  1.97E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419024BDBM50419024(CHEMBL1814300)
Affinity DataEC50:  2.20E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419026BDBM50419026(CHEMBL231391)
Affinity DataEC50:  2.37E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419023BDBM50419023(CHEMBL1814305)
Affinity DataEC50:  2.50E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50295926BDBM50295926(Magreth-14a | 5,3'-Diallyl-4'-methoxy-biphenyl-2-o...)
Affinity DataEC50:  2.72E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419029BDBM50419029(CHEMBL1814291)
Affinity DataEC50:  3.42E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419027BDBM50419027(CHEMBL182529)
Affinity DataEC50:  3.52E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 78304BDBM78304(2-(2-hydroxy-5-prop-2-enylphenyl)-4-prop-2-enylphe...)
Affinity DataEC50:  3.68E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157304BDBM50157304(3',5-diallylbiphenyl-2,4'-diol | CHEMBL16901 | cid...)
Affinity DataEC50:  3.93E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50295927BDBM50295927(5,3'-Diallyl-2,4'-dimethoxy-biphenyl | 2,4'-Dimeth...)
Affinity DataEC50:  4.21E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419025BDBM50419025(CHEMBL1814295)
Affinity DataEC50:  5.43E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81564BDBM81564(Magreth-16b)
Affinity DataEC50:  5.99E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Human)
University of Vienna

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419028BDBM50419028(CHEMBL1814293)
Affinity DataEC50:  1.05E+5nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed