Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50001228
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013943BDBM50013943(CHEMBL327270 | Furan-2-carboxylic acid (2-chloro-p...)
Affinity DataKi:  0.130nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013945BDBM50013945(CHEMBL431047 | Furan-2-carboxylic acid [3-methyl-1...)
Affinity DataKi:  0.150nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013934BDBM50013934(CHEMBL319060 | N-(2-Fluoro-phenyl)-2-methoxy-N-(3-...)
Affinity DataKi:  0.190nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013934BDBM50013934(CHEMBL319060 | N-(2-Fluoro-phenyl)-2-methoxy-N-(3-...)
Affinity DataKi:  0.190nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 94503BDBM94503(N-[4-(methoxymethyl)-1-(2-thiophen-2-ylethyl)piper...)
Affinity DataKi:  0.220nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013939BDBM50013939(CHEMBL95247 | Furan-2-carboxylic acid (3-methyl-1-...)
Affinity DataKi:  0.300nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013939BDBM50013939(CHEMBL95247 | Furan-2-carboxylic acid (3-methyl-1-...)
Affinity DataKi:  0.300nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013938BDBM50013938(CHEMBL318958 | 2-Methoxy-N-(3-methyl-1-phenethyl-p...)
Affinity DataKi:  0.330nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013938BDBM50013938(CHEMBL318958 | 2-Methoxy-N-(3-methyl-1-phenethyl-p...)
Affinity DataKi:  0.330nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013949BDBM50013949(CHEMBL95248 | Furan-2-carboxylic acid (2-methoxy-p...)
Affinity DataKi:  0.780nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013948BDBM50013948(CHEMBL95909 | N-(2-Chloro-phenyl)-2-methoxy-N-(3-m...)
Affinity DataKi:  1.10nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013935BDBM50013935(CHEMBL95390 | N-(2-Fluoro-phenyl)-2-methoxy-N-[3-m...)
Affinity DataKi:  2nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013947BDBM50013947(CHEMBL95786 | Furan-2-carboxylic acid (2-methoxy-p...)
Affinity DataKi:  2nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000092BDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataKi:  2.10nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50008984BDBM50008984(N-(1-Phenethyl-piperidin-4-yl)-N-phenyl-propionami...)
Affinity DataKi:  2.20nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013940BDBM50013940(CHEMBL319343 | N-(2-Fluoro-phenyl)-2-methoxy-N-[3-...)
Affinity DataKi:  2.20nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013942BDBM50013942(CHEMBL318895 | N-(2-Chloro-phenyl)-2-methoxy-N-(3-...)
Affinity DataKi:  2.80nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013936BDBM50013936(CHEMBL100111 | 2-Methoxy-N-(3-methyl-1-phenethyl-p...)
Affinity DataKi:  4.20nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013936BDBM50013936(CHEMBL100111 | 2-Methoxy-N-(3-methyl-1-phenethyl-p...)
Affinity DataKi:  4.20nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013944BDBM50013944(CHEMBL329950 | 2-Methoxy-N-(2-methoxy-phenyl)-N-(3...)
Affinity DataKi:  7.60nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013941BDBM50013941(CHEMBL99596 | N-(2-Fluoro-phenyl)-2-methoxy-N-(3-m...)
Affinity DataKi:  8.10nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 83450BDBM83450(N-[1-[2-(4-ethyl-5-oxidanylidene-1,2,3,4-tetrazol-...)
Affinity DataKi:  8.20nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013937BDBM50013937(CHEMBL317822 | 2-Methoxy-N-(2-methoxy-phenyl)-N-[3...)
Affinity DataKi:  11nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013946BDBM50013946(CHEMBL316670 | Furan-2-carboxylic acid (2-methoxy-...)
Affinity DataKi: >100nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013935BDBM50013935(CHEMBL95390 | N-(2-Fluoro-phenyl)-2-methoxy-N-[3-m...)
Affinity DataKi: >1.00E+3nMAssay Description:Ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed