Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 8175
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 7.30E+3nMAssay Description:The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM235705(L-Isoseryl-L-phenylalanyl-L-leucine hydrochloride ...)
Affinity DataIC50: 1.22E+4nMAssay Description:The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM235704(L-Isoseryl-L-leucyl-L-phenylalanine hydrochloride ...)
Affinity DataIC50: 2.09E+4nMAssay Description:The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM235703(L-Isoseryl-L-phenylalanyl-L-leucine benzyl ester h...)
Affinity DataIC50: 3.22E+4nMAssay Description:The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM235701(L-Isoseryl-L-phenylalanyl-L-leucine methyl ester h...)
Affinity DataIC50: 6.51E+4nMAssay Description:The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM235702(L-Isoseryl-L-leucyl-L-phenylalanine benzyl ester h...)
Affinity DataIC50: 6.91E+4nMAssay Description:The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM235697(L-Isoseryl-L- phenylalanine benzyl ester hydrochlo...)
Affinity DataIC50: 9.95E+4nMAssay Description:The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

LigandPNGBDBM235704(L-Isoseryl-L-leucyl-L-phenylalanine hydrochloride ...)
Affinity DataIC50: 1.15E+5nMpH: 8.5 T: 2°CAssay Description:The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

LigandPNGBDBM235700(L-Isoseryl-L-leucyl-L-phenylalanine methyl ester h...)
Affinity DataIC50: 1.26E+5nMpH: 8.5 T: 2°CAssay Description:The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM235700(L-Isoseryl-L-leucyl-L-phenylalanine methyl ester h...)
Affinity DataIC50: 1.40E+5nMAssay Description:The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 1.67E+5nMpH: 8.5 T: 2°CAssay Description:The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM235698(L-Isoseryl-L-leucine benzyl ester hydrochloride (1...)
Affinity DataIC50: 1.95E+5nMAssay Description:The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM50010209(CHEMBL3251694 | L-Isoseryl-L-leucine hydrochloride...)
Affinity DataIC50: 1.99E+5nMAssay Description:The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

LigandPNGBDBM235705(L-Isoseryl-L-phenylalanyl-L-leucine hydrochloride ...)
Affinity DataIC50: 2.03E+5nMpH: 8.5 T: 2°CAssay Description:The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

LigandPNGBDBM235701(L-Isoseryl-L-phenylalanyl-L-leucine methyl ester h...)
Affinity DataIC50: 2.25E+5nMpH: 8.5 T: 2°CAssay Description:The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM235696(L-Isoseryl-L-leucine methyl ester hydrochloride (1...)
Affinity DataIC50: 2.29E+5nMAssay Description:The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

LigandPNGBDBM235702(L-Isoseryl-L-leucyl-L-phenylalanine benzyl ester h...)
Affinity DataIC50: 2.37E+5nMpH: 8.5 T: 2°CAssay Description:The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM235699((2S)-2-[(2S)-3-amino-2-hydroxypropanamido]-3-pheny...)
Affinity DataIC50: 2.49E+5nMAssay Description:The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM235695(Methyl (2S)-2-[(2S)-3-amino-2-hydroxypropanamido]-...)
Affinity DataIC50: 3.02E+5nMAssay Description:The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

LigandPNGBDBM235697(L-Isoseryl-L- phenylalanine benzyl ester hydrochlo...)
Affinity DataIC50: 3.29E+5nMpH: 8.5 T: 2°CAssay Description:The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

LigandPNGBDBM235703(L-Isoseryl-L-phenylalanyl-L-leucine benzyl ester h...)
Affinity DataIC50: 3.34E+5nMpH: 8.5 T: 2°CAssay Description:The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

LigandPNGBDBM50010209(CHEMBL3251694 | L-Isoseryl-L-leucine hydrochloride...)
Affinity DataIC50: 3.64E+5nMpH: 8.5 T: 2°CAssay Description:The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

LigandPNGBDBM235696(L-Isoseryl-L-leucine methyl ester hydrochloride (1...)
Affinity DataIC50: 6.82E+5nMpH: 8.5 T: 2°CAssay Description:The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

LigandPNGBDBM235699((2S)-2-[(2S)-3-amino-2-hydroxypropanamido]-3-pheny...)
Affinity DataIC50: 7.10E+5nMpH: 8.5 T: 2°CAssay Description:The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

LigandPNGBDBM235698(L-Isoseryl-L-leucine benzyl ester hydrochloride (1...)
Affinity DataIC50: 1.00E+6nMpH: 8.5 T: 2°CAssay Description:The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

LigandPNGBDBM235695(Methyl (2S)-2-[(2S)-3-amino-2-hydroxypropanamido]-...)
Affinity DataIC50: 1.00E+6nMpH: 8.5 T: 2°CAssay Description:The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details Article
PubMed