Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50033871
TargetAndrogen receptor(Human)
University of British Columbia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353034BDBM50353034(CHEMBL1302748)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human AR AF2 site expressed in human LNCap cells coexpressing eGFP -ARR2PB assessed as inhibition of transcriptional activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of British Columbia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353033BDBM50353033(CHEMBL1527972)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of human AR AF2 site expressed in human LNCap cells coexpressing eGFP -ARR2PB assessed as inhibition of transcriptional activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of British Columbia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353035BDBM50353035(CHEMBL1822155)
Affinity DataIC50: 8.20E+3nMAssay Description:Displacement of SRC2-3 peptide from human AR ligand binding site expressed in Escherichia coli BL21 by AF2 FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of British Columbia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 33070BDBM33070(MLS000068595 | cid_760604 | SMR000122974 | 4-(2,3-...)
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of human AR AF2 site expressed in human LNCap cells coexpressing eGFP -ARR2PB assessed as inhibition of transcriptional activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of British Columbia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353036BDBM50353036(CHEMBL1822156)
Affinity DataIC50: 1.86E+4nMAssay Description:Inhibition of human AR AF2 site expressed in human LNCap cells coexpressing eGFP -ARR2PB assessed as inhibition of transcriptional activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of British Columbia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353037BDBM50353037(CHEMBL1822157)
Affinity DataIC50: 2.60E+4nMAssay Description:Displacement of SRC2-3 peptide from human AR ligand binding site expressed in Escherichia coli BL21 by AF2 FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of British Columbia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353036BDBM50353036(CHEMBL1822156)
Affinity DataIC50: 3.06E+4nMAssay Description:Displacement of SRC2-3 peptide from human AR ligand binding site expressed in Escherichia coli BL21 by AF2 FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of British Columbia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353033BDBM50353033(CHEMBL1527972)
Affinity DataIC50: 3.07E+4nMAssay Description:Displacement of SRC2-3 peptide from human AR ligand binding site expressed in Escherichia coli BL21 by AF2 FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of British Columbia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 33070BDBM33070(MLS000068595 | cid_760604 | SMR000122974 | 4-(2,3-...)
Affinity DataIC50: 3.15E+4nMAssay Description:Displacement of SRC2-3 peptide from human AR ligand binding site expressed in Escherichia coli BL21 by AF2 FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of British Columbia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353034BDBM50353034(CHEMBL1302748)
Affinity DataIC50: 3.29E+4nMAssay Description:Displacement of SRC2-3 peptide from human AR ligand binding site expressed in Escherichia coli BL21 by AF2 FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of British Columbia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353037BDBM50353037(CHEMBL1822157)
Affinity DataIC50: 3.34E+4nMAssay Description:Inhibition of human AR AF2 site expressed in human LNCap cells coexpressing eGFP -ARR2PB assessed as inhibition of transcriptional activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of British Columbia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353035BDBM50353035(CHEMBL1822155)
Affinity DataIC50: 3.44E+4nMAssay Description:Inhibition of human AR AF2 site expressed in human LNCap cells coexpressing eGFP -ARR2PB assessed as inhibition of transcriptional activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed