Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50033915
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti���Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099491BDBM50099491(cid_3392731 | CHEMBL21241 | 2-(4-{2-[3-Cyclohexyl-...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at Gal4-fused PPARalpha expressed in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti���Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353757BDBM50353757(CHEMBL1828826)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at Gal4-fused PPARalpha expressed in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti���Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353755BDBM50353755(CHEMBL1828822)
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at Gal4-fused PPARalpha expressed in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti���Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353751BDBM50353751(CHEMBL1828831)
Affinity DataEC50:  9.10E+3nMAssay Description:Agonist activity at Gal4-fused PPARalpha expressed in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti���Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353752BDBM50353752(CHEMBL1828832)
Affinity DataEC50:  9.30E+3nMAssay Description:Agonist activity at Gal4-fused PPARalpha expressed in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti���Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353750BDBM50353750(CHEMBL19641)
Affinity DataEC50:  9.30E+3nMAssay Description:Agonist activity at Gal4-fused PPARalpha expressed in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti���Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353754BDBM50353754(CHEMBL1828821)
Affinity DataEC50:  1.13E+4nMAssay Description:Agonist activity at Gal4-fused PPARalpha expressed in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti���Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353756BDBM50353756(CHEMBL1828825)
Affinity DataEC50:  1.88E+4nMAssay Description:Agonist activity at Gal4-fused PPARalpha expressed in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti���Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353749BDBM50353749(CHEMBL1828829)
Affinity DataEC50:  2.71E+4nMAssay Description:Agonist activity at Gal4-fused PPARalpha expressed in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti���Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353753BDBM50353753(CHEMBL1828834)
Affinity DataEC50:  4.37E+4nMAssay Description:Agonist activity at Gal4-fused PPARalpha expressed in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti���Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110590BDBM50110590(5-(2,5-dimethylphenoxy)-2,2-dimethylpentanoic acid...)
Affinity DataEC50:  5.90E+4nMAssay Description:Agonist activity at Gal4-fused PPARalpha expressed in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti���Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353759BDBM50353759(CHEMBL1828828)
Affinity DataEC50:  6.15E+4nMAssay Description:Agonist activity at Gal4-fused PPARalpha expressed in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti���Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353758BDBM50353758(CHEMBL1828827)
Affinity DataEC50:  1.09E+5nMAssay Description:Agonist activity at Gal4-fused PPARalpha expressed in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed