Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50034034
TargetAmine oxidase [flavin-containing] A(Human)
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 30.2nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells assessed as inhibition of kynuramine oxidation after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAmine oxidase [flavin-containing] B(Human)
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 85.2nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells assessed as inhibition of kynuramine oxidation after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM50355808(CHEMBL1911928)
Affinity DataIC50: 171nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells assessed as inhibition of kynuramine oxidation after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM50355807(CHEMBL1911927)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells assessed as inhibition of kynuramine oxidation after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM50355806(CHEMBL1911926)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect cells assessed as inhibition of kynuramine oxidation after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM50355808(CHEMBL1911928)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human recombinant MAO-A expressed in insect cells assessed as inhibition of kynuramine oxidation after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed