Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50034095
LigandPNGBDBM50356930(CHEMBL1914475)
Affinity DataIC50: 25nMAssay Description:Inhibition of PI3Kalpha by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50189744((Z)-5-((5-(4-fluoro-2-hydroxyphenyl)furan-2-yl)met...)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human PI3Kgamma by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50356930(CHEMBL1914475)
Affinity DataIC50: 34nMAssay Description:Inhibition of recombinant human PI3Kgamma by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50356940(CHEMBL1916047)
Affinity DataIC50: 230nMAssay Description:Inhibition of recombinant human PI3Kgamma by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50356930(CHEMBL1914475)
Affinity DataIC50: 760nMAssay Description:Inhibition of PI3Kgamma in human neutrophils assessed as inhibition of fMLP-stimulated superoxide productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50356939(CHEMBL1916046)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of recombinant human PI3Kgamma by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50356937(CHEMBL1728139)
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of recombinant human PI3Kgamma assessed as depletion of ATP by kinase-glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50356931(CHEMBL1916042)
Affinity DataIC50: 1.56E+5nMAssay Description:Inhibition of recombinant human PI3Kgamma assessed as depletion of ATP by kinase-glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50356932(CHEMBL1889525 | cid_40237)
Affinity DataIC50: 3.80E+5nMAssay Description:Inhibition of recombinant human PI3Kgamma assessed as depletion of ATP by kinase-glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50356935(CHEMBL1916044)
Affinity DataIC50: 3.95E+5nMAssay Description:Inhibition of recombinant human PI3Kgamma assessed as depletion of ATP by kinase-glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50356936(CHEMBL1916045)
Affinity DataIC50: 7.73E+5nMAssay Description:Inhibition of recombinant human PI3Kgamma assessed as depletion of ATP by kinase-glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50356938(CHEMBL1916048)
Affinity DataIC50: 9.15E+5nMAssay Description:Inhibition of recombinant human PI3Kgamma assessed as depletion of ATP by kinase-glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50356933(CHEMBL1887078)
Affinity DataIC50: 1.60E+6nMAssay Description:Inhibition of recombinant human PI3Kgamma assessed as depletion of ATP by kinase-glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50356934(CHEMBL1916043)
Affinity DataIC50: 1.67E+6nMAssay Description:Inhibition of recombinant human PI3Kgamma assessed as depletion of ATP by kinase-glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed