Found 14 Enz. Inhib. hit(s) with all data for entry = 50034117 TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of rat Nav1.2 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
Affinity DataIC50: 3.96E+4nMAssay Description:Inhibition of mouse Nav1.6 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by t...More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 5.23E+4nMAssay Description:Inhibition of rat Nav1.2 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Rattus norvegicus (Rat))
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 5.43E+4nMAssay Description:Inhibition of rat Nav1.4 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
Affinity DataIC50: 5.43E+4nMAssay Description:Inhibition of mouse Nav1.6 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by t...More data for this Ligand-Target Pair
TargetSodium channel protein type 3 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of rat Nav1.3 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 1 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 1.74E+5nMAssay Description:Inhibition of rat Nav1.1 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 1.77E+5nMAssay Description:Inhibition of rat Nav1.7 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Rattus norvegicus (Rat))
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 2.04E+5nMAssay Description:Inhibition of rat Nav1.4 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 2.37E+5nMAssay Description:Inhibition of rat Nav1.5 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat Nav1.7 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 3 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat Nav1.3 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 1 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat Nav1.1 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 8.71E+5nMAssay Description:Inhibition of rat Nav1.5 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
