Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50034211
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358895BDBM50358895(CHEMBL1923571)
Affinity DataIC50: 0.170nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353052BDBM50353052(CHEMBL1822515)
Affinity DataIC50: 0.190nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353052BDBM50353052(CHEMBL1822515)
Affinity DataIC50: 0.190nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358897BDBM50358897(CHEMBL1923573)
Affinity DataIC50: 0.230nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358912BDBM50358912(CHEMBL1923588)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358909BDBM50358909(CHEMBL1923585)
Affinity DataIC50: 0.330nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358899BDBM50358899(CHEMBL1923575)
Affinity DataIC50: 0.350nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358907BDBM50358907(CHEMBL1923583)
Affinity DataIC50: 0.350nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358904BDBM50358904(CHEMBL1923580)
Affinity DataIC50: 0.360nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358914BDBM50358914(CHEMBL1923590)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358913BDBM50358913(CHEMBL1923589)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358898BDBM50358898(CHEMBL1923574)
Affinity DataIC50: 0.470nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358893BDBM50358893(CHEMBL1923594)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358908BDBM50358908(CHEMBL1923584)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358894BDBM50358894(CHEMBL1923570)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358903BDBM50358903(CHEMBL1923579)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358901BDBM50358901(CHEMBL1923577)
Affinity DataIC50: 0.540nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358891BDBM50358891(CHEMBL1923593)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358900BDBM50358900(CHEMBL1923576)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358890BDBM50358890(CHEMBL1923592)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358902BDBM50358902(CHEMBL1923578)
Affinity DataIC50: 1nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358910BDBM50358910(CHEMBL1923586)
Affinity DataIC50: 1nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358906BDBM50358906(CHEMBL1923582)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358916BDBM50358916(CHEMBL1923569)
Affinity DataIC50: 1.14nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358911BDBM50358911(CHEMBL1923587)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358892BDBM50358892(CHEMBL1921819)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353039BDBM50353039(CHEMBL1821735)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358896BDBM50358896(CHEMBL1923572)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358905BDBM50358905(CHEMBL1923581)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353046BDBM50353046(CHEMBL1822525)
Affinity DataIC50: 9nMAssay Description:Inhibition of human GST-tagged ALK expressed in SF21 insect cells using PLCgamma/GST as substrate after 15 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358916BDBM50358916(CHEMBL1923569)
Affinity DataIC50: 30nMAssay Description:Inhibition of human GST-tagged ALK expressed in SF21 insect cells using PLCgamma/GST as substrate after 15 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353046BDBM50353046(CHEMBL1822525)
Affinity DataIC50: 379nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Cephalon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50358915BDBM50358915(CHEMBL1923591)
Affinity DataIC50: 480nMAssay Description:Inhibition of human recombinant JAK2 using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed