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Found 12 Enz. Inhib. hit(s) with all data for entry = 50034394
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50361661(CHEMBL1940484)
Affinity DataKi:  437nMAssay Description:Displacement of [3H](+)pentazocine from sigma 1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50361658(CHEMBL1940482)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)pentazocine from sigma 1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50361660(CHEMBL1940599)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)pentazocine from sigma 1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50276978(1-(4-benzylpiperidin-1-yl)-2-(5-hydroxy-1Hindol-3-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)pentazocine from sigma 1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50276976(2-(4-benzylpiperidin-1-yl)-1-(5-hydroxy-1Hindol-3-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)pentazocine from sigma 1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50361658(CHEMBL1940482)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]ifenprodil from GluN2B/NMDA in Wistar rat cerebral cortex after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50361660(CHEMBL1940599)
Affinity DataIC50:  22nMAssay Description:Displacement of [3H]ifenprodil from GluN2B/NMDA in Wistar rat cerebral cortex after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50361654(CHEMBL1940477)
Affinity DataIC50:  324nMAssay Description:Displacement of [3H]ifenprodil from GluN2B/NMDA in Wistar rat cerebral cortex after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50361659(CHEMBL1940597)
Affinity DataIC50:  1.99E+3nMAssay Description:Displacement of [3H]ifenprodil from GluN2B/NMDA in Wistar rat cerebral cortex after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50361656(CHEMBL1940479)
Affinity DataIC50:  2.91E+3nMAssay Description:Displacement of [3H]ifenprodil from GluN2B/NMDA in Wistar rat cerebral cortex after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50361655(CHEMBL1940478)
Affinity DataIC50:  6.64E+3nMAssay Description:Displacement of [3H]ifenprodil from GluN2B/NMDA in Wistar rat cerebral cortex after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50361657(CHEMBL1940480)
Affinity DataIC50:  7.14E+3nMAssay Description:Displacement of [3H]ifenprodil from GluN2B/NMDA in Wistar rat cerebral cortex after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed