Compile Data Set for Download or QSAR
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Found 26 Enz. Inhib. hit(s) with all data for entry = 50034337
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360782(CHEMBL1934513)
Affinity DataIC50:  25nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360774(CHEMBL1934647)
Affinity DataIC50:  103nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360779(CHEMBL1934516)
Affinity DataIC50:  111nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360780(CHEMBL1934515)
Affinity DataIC50:  202nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360785(CHEMBL1934508)
Affinity DataIC50:  212nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360781(CHEMBL1934514)
Affinity DataIC50:  271nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360771(CHEMBL1934650)
Affinity DataIC50:  327nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360773(CHEMBL1934648)
Affinity DataIC50:  332nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360775(CHEMBL1934646)
Affinity DataIC50:  546nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360778(CHEMBL1934641)
Affinity DataIC50:  685nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360769(CHEMBL1934652)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360772(CHEMBL1934649)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360776(CHEMBL1934645)
Affinity DataIC50:  2.03E+3nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360770(CHEMBL1934651)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360789(CHEMBL1934503)
Affinity DataIC50:  3.82E+3nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360794(CHEMBL1934497)
Affinity DataIC50:  4.74E+3nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360787(CHEMBL1934505)
Affinity DataIC50:  6.88E+3nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360791(CHEMBL1934501)
Affinity DataIC50:  7.91E+3nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360788(CHEMBL1934504)
Affinity DataIC50:  9.64E+3nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360790(CHEMBL1934502)
Affinity DataIC50:  9.75E+3nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360777(CHEMBL1934644)
Affinity DataIC50:  1.01E+4nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360783(CHEMBL1934510)
Affinity DataIC50:  1.17E+4nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360784(CHEMBL1934509)
Affinity DataIC50:  1.39E+4nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360786(CHEMBL1934506)
Affinity DataIC50:  1.45E+4nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360792(CHEMBL1934499)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50360793(CHEMBL1934498)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of B-Raf in human A375 cells assessed as inhibition of phosphorylation of MEK1/2 by meso scale assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed