Compile Data Set for Download or QSAR
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Found 17 Enz. Inhib. hit(s) with all data for entry = 50034284
TargetSphingosine kinase 2(Mus musculus (Mouse))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359977(CHEMBL1927590)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of mouse SphK2 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Mus musculus (Mouse))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359976(CHEMBL1927588)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of mouse SphK2 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Mus musculus (Mouse))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359979(CHEMBL1927596)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of mouse SphK2 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359980(CHEMBL1927600)
Affinity DataKi:  1.65E+4nMAssay Description:Inhibition of SphK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359973(CHEMBL1927579)
Affinity DataKi:  2.20E+4nMAssay Description:Inhibition of human SphK1 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Mus musculus (Mouse))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359975(CHEMBL1927583)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibition of mouse SphK2 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Mus musculus (Mouse))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359974(CHEMBL1927581)
Affinity DataKi:  2.90E+4nMAssay Description:Inhibition of mouse SphK2 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359974(CHEMBL1927581)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of human SphK1 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Mus musculus (Mouse))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359978(CHEMBL1927592)
Affinity DataKi:  3.30E+4nMAssay Description:Inhibition of mouse SphK2 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Mus musculus (Mouse))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359973(CHEMBL1927579)
Affinity DataKi:  3.80E+4nMAssay Description:Inhibition of mouse SphK2 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Mus musculus (Mouse))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359972(CHEMBL1927562)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of mouse SphK2 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359975(CHEMBL1927583)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of human SphK1 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359977(CHEMBL1927590)
Affinity DataKi:  4.70E+4nMAssay Description:Inhibition of human SphK1 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359976(CHEMBL1927588)
Affinity DataKi:  6.00E+4nMAssay Description:Inhibition of human SphK1 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359979(CHEMBL1927596)
Affinity DataKi:  7.00E+4nMAssay Description:Inhibition of human SphK1 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359972(CHEMBL1927562)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human SphK1 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50359978(CHEMBL1927592)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human SphK1 expressed in baculovirus infected Sf9 insect cells using sphingosine and [gamma-(32)P]-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed