Compile Data Set for Download or QSAR
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Found 8 Enz. Inhib. hit(s) with all data for entry = 50039508
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50305083(3-((3S,6S)-6-Isobutyl-9-methoxy-1,4-dioxo-1,2,3,4,...)
Affinity DataIC50:  50nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50379211(CHEMBL2011288)
Affinity DataIC50:  110nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50379213(CHEMBL2011290)
Affinity DataIC50:  160nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50379209(CHEMBL2011282)
Affinity DataIC50:  170nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50379208(CHEMBL2011287)
Affinity DataIC50:  180nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50379212(CHEMBL2011289)
Affinity DataIC50:  200nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50379210(CHEMBL2011286)
Affinity DataIC50:  470nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50305083(3-((3S,6S)-6-Isobutyl-9-methoxy-1,4-dioxo-1,2,3,4,...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of MRP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed