Compile Data Set for Download or QSAR
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Found 29 Enz. Inhib. hit(s) with all data for entry = 50034423
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362167(CHEMBL1941129)
Affinity DataIC50:  5.5nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362160(CHEMBL1941121)
Affinity DataIC50:  5.80nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362159(CHEMBL1941120)
Affinity DataIC50:  6.20nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362158(CHEMBL1941119)
Affinity DataIC50:  9.20nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362166(CHEMBL1941128)
Affinity DataIC50:  9.70nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362164(CHEMBL1941126)
Affinity DataIC50:  11nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362157(CHEMBL1941118)
Affinity DataIC50:  11nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362165(CHEMBL1941127)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362167(CHEMBL1941129)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362162(CHEMBL1941123)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362156(CHEMBL1941117)
Affinity DataIC50:  18nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362166(CHEMBL1941128)
Affinity DataIC50:  18nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362155(CHEMBL1941116)
Affinity DataIC50:  42nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362165(CHEMBL1941127)
Affinity DataIC50:  52nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362161(CHEMBL1941122)
Affinity DataIC50:  99nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362164(CHEMBL1941126)
Affinity DataIC50:  99nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362162(CHEMBL1941123)
Affinity DataIC50:  128nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362156(CHEMBL1941117)
Affinity DataIC50:  147nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362160(CHEMBL1941121)
Affinity DataIC50:  211nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362155(CHEMBL1941116)
Affinity DataIC50:  256nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362157(CHEMBL1941118)
Affinity DataIC50:  359nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362163(CHEMBL1941124)
Affinity DataIC50:  502nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362159(CHEMBL1941120)
Affinity DataIC50:  772nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362161(CHEMBL1941122)
Affinity DataIC50:  797nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362163(CHEMBL1941124)
Affinity DataIC50:  990nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362168(CHEMBL1941125)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362155(CHEMBL1941116)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]PGD2 from human DP1 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Cavia porcellus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362158(CHEMBL1941119)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]PGD2 from guinea pig CRTH2 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50362165(CHEMBL1941127)
Affinity DataIC50:  5.20E+3nMAssay Description:Displacement of [3H]PGD2 from human DP1 receptor expressed in HEK293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed