Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50022591
Affinity DataKd: 1.5nMAssay Description:Inhibition of non-phosphorylated human N-terminal His-P38alpha overexpressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by Kino...More data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human p38alpha using ATF2 as substrate in presence of 33P-ATP by ProQinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of activated human P38alphaMore data for this Ligand-Target Pair
Affinity DataKd: 7.60nMAssay Description:Inhibition of non-phosphorylated human N-terminal His-P38alpha overexpressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by Kino...More data for this Ligand-Target Pair
3D Structure (crystal)TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Tubingen
Curated by ChEMBL
University of Tubingen
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of p38-MAPK in human HeLa cells assessed as HSP27 phosphorylation at Ser82 level incubated for 2 hrs in the presence of anisomycin stimula...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of P38alpha in human THP-1 cells incubated for 30 mins by whole blood assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of non-phosphorylated human N-terminal His-P38alpha overexpressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of P38alpha in human THP-1 cells incubated for 30 mins by whole blood assayMore data for this Ligand-Target Pair
