Compile Data Set for Download or QSAR
maximum 50k data
Found 79 Enz. Inhib. hit(s) with all data for entry = 50041969
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419792(CHEMBL1950609)
Affinity DataIC50:  1.70E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419827(CHEMBL1950506)
Affinity DataIC50:  2.40E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419851(CHEMBL1950510)
Affinity DataIC50:  2.82E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419806(CHEMBL1950626)
Affinity DataIC50:  2.88E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419789(CHEMBL1950606)
Affinity DataIC50:  3.89E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419816(CHEMBL1950637)
Affinity DataIC50:  3.90E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419796(CHEMBL1950614)
Affinity DataIC50:  4.17E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419829(CHEMBL1950508)
Affinity DataIC50:  4.27E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419814(CHEMBL1950635)
Affinity DataIC50:  4.30E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419848(CHEMBL1950622)
Affinity DataIC50:  4.47E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419802(CHEMBL1949684)
Affinity DataIC50:  4.47E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50149054(2-(3,3-Dimethyl-2,5-dioxo-pyrrolidin-1-yl)-benzoic...)
Affinity DataIC50:  4.90E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50149051(2-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-benzoic ac...)
Affinity DataIC50:  5.01E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419803(CHEMBL1950623)
Affinity DataIC50:  5.13E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419798(CHEMBL1950616)
Affinity DataIC50:  5.13E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419842(CHEMBL465057)
Affinity DataIC50:  5.37E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50149044(2-Acetylamino-benzoic acid 1-(3-phenyl-propyl)-pip...)
Affinity DataIC50:  5.50E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419815(CHEMBL1950636)
Affinity DataIC50:  5.60E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419839(CHEMBL1950522)
Affinity DataIC50:  5.62E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419817(CHEMBL1950638)
Affinity DataIC50:  5.90E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419815(CHEMBL1950636)
Affinity DataIC50:  6.03E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50149039(Biphenyl-4-carboxylic acid 1-(3-phenyl-propyl)-pip...)
Affinity DataIC50:  6.31E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419830(CHEMBL1950509)
Affinity DataIC50:  6.46E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419821(CHEMBL1950639)
Affinity DataIC50:  6.50E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419809(CHEMBL1950630)
Affinity DataIC50:  6.90E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419850(CHEMBL1950505)
Affinity DataIC50:  6.92E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419826(CHEMBL1950504)
Affinity DataIC50:  7.08E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419841(CHEMBL1950600)
Affinity DataIC50:  7.08E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419791(CHEMBL1950608)
Affinity DataIC50:  7.24E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419790(CHEMBL1950607)
Affinity DataIC50:  7.41E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419808(CHEMBL1950629)
Affinity DataIC50:  7.50E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419834(CHEMBL1950515)
Affinity DataIC50:  7.59E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50149043(2-Trifluoromethyl-benzoic acid 1-(3-phenyl-propyl)...)
Affinity DataIC50:  7.94E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50149050(2-Methoxy-benzoic acid 1-(3-phenyl-propyl)-piperid...)
Affinity DataIC50:  7.94E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50149043(2-Trifluoromethyl-benzoic acid 1-(3-phenyl-propyl)...)
Affinity DataIC50:  8.00E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419805(CHEMBL1950625)
Affinity DataIC50:  8.10E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419805(CHEMBL1950625)
Affinity DataIC50:  8.13E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419799(CHEMBL1950618)
Affinity DataIC50:  8.32E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419800(CHEMBL1950619)
Affinity DataIC50:  8.71E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419853(CHEMBL1950521)
Affinity DataIC50:  8.91E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419847(CHEMBL1950617)
Affinity DataIC50:  8.91E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419828(CHEMBL1950507)
Affinity DataIC50:  9.12E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50149041(2-Chloro-benzoic acid 1-(3-phenyl-propyl)-piperidi...)
Affinity DataIC50:  9.33E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419832(CHEMBL1950513)
Affinity DataIC50:  9.55E+3nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419823(CHEMBL1950501)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419822(CHEMBL1950500)
Affinity DataIC50:  1.02E+4nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419838(CHEMBL1950520)
Affinity DataIC50:  1.05E+4nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419813(CHEMBL1950634)
Affinity DataIC50:  1.07E+4nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419797(CHEMBL1950615)
Affinity DataIC50:  1.07E+4nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50419831(CHEMBL1950512)
Affinity DataIC50:  1.10E+4nMAssay Description:Antagonist activity at human nAChR alpha4/beta2 receptor expressed in HEK ts201 cells assessed as calcium accumulation by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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