Compile Data Set for Download or QSAR
maximum 50k data
Found 33 Enz. Inhib. hit(s) with all data for entry = 50039520
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379308(CHEMBL2011816)
Affinity DataKi:  4.40nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379328(CHEMBL2011825)
Affinity DataIC50:  0.200nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379309(CHEMBL2011826)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379312(CHEMBL2011892)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379320(CHEMBL2011834)
Affinity DataIC50:  2.5nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379322(CHEMBL2011832)
Affinity DataIC50:  2.5nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379310(CHEMBL2011894)
Affinity DataIC50:  3nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379334(CHEMBL2011819)
Affinity DataIC50:  3nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379319(CHEMBL2011835)
Affinity DataIC50:  4.10nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379314(CHEMBL2011890)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379311(CHEMBL2011893)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379308(CHEMBL2011816)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at mouse GHSR1 receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379335(CHEMBL2011818)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379323(CHEMBL2011831)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50153547(3-(2,6-Dichloro-phenyl)-5-[2-(2-oxo-piperidin-1-yl...)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as blockade of intracellular Ca2+ mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379308(CHEMBL2011816)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379336(CHEMBL2011817)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379326(CHEMBL2011828)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50158327((+/-)isobutyl 2-((4-(diethylamino)phenyl)carbamoyl...)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as blockade of intracellular Ca2+ mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379321(CHEMBL2011833)
Affinity DataIC50:  16.5nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379313(CHEMBL2011891)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379331(CHEMBL2011822)
Affinity DataIC50:  26nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379332(CHEMBL2011821)
Affinity DataIC50:  28nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379317(CHEMBL2011887)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379329(CHEMBL2011824)
Affinity DataIC50:  79nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379330(CHEMBL2011823)
Affinity DataIC50:  143nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379333(CHEMBL2011820)
Affinity DataIC50:  171nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379325(CHEMBL2011829)
Affinity DataIC50:  196nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379318(CHEMBL2011836)
Affinity DataIC50:  313nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379327(CHEMBL2011827)
Affinity DataIC50:  314nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379324(CHEMBL2011830)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379316(CHEMBL2011888)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379315(CHEMBL2011889)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed