Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50039523
TargetAndrogen receptor(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50379430(CHEMBL1802077)
Affinity DataIC50:  600nMAssay Description:Antagonist activity at androgen receptor in human LNCAP cells assessed as decrease in prostate specific antigen mRNA level after 20 hrs by real time ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50379430(CHEMBL1802077)
Affinity DataIC50:  750nMAssay Description:Antagonist activity at androgen receptor in human LNCAP cells assessed as decrease in transmembrane protease serine 2 mRNA level after 20 hrs by real...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed