Compile Data Set for Download or QSAR
maximum 50k data
Found 42 Enz. Inhib. hit(s) with all data for entry = 50039750
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383311(CHEMBL2029619)
Affinity DataIC50:  40nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383305(CHEMBL2029615)
Affinity DataIC50:  50nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383306(CHEMBL2029618)
Affinity DataIC50:  90nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383304(CHEMBL2029622)
Affinity DataIC50:  270nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  300nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383304(CHEMBL2029622)
Affinity DataIC50:  520nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383306(CHEMBL2029618)
Affinity DataIC50:  570nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383311(CHEMBL2029619)
Affinity DataIC50:  670nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383307(CHEMBL2029614)
Affinity DataIC50:  950nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383312(CHEMBL2029620)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383306(CHEMBL2029618)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383305(CHEMBL2029615)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383313(CHEMBL2029623)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383305(CHEMBL2029615)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383308(CHEMBL523951)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383306(CHEMBL2029618)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383305(CHEMBL2029615)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383307(CHEMBL2029614)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383308(CHEMBL523951)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383309(CHEMBL2029616)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383310(BUCHENAVIANINE)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383304(CHEMBL2029622)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383305(CHEMBL2029615)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383312(CHEMBL2029620)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383304(CHEMBL2029622)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383310(BUCHENAVIANINE)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383307(CHEMBL2029614)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383305(CHEMBL2029615)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383308(CHEMBL523951)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383309(CHEMBL2029616)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383310(BUCHENAVIANINE)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383311(CHEMBL2029619)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383312(CHEMBL2029620)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383304(CHEMBL2029622)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383313(CHEMBL2029623)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383309(CHEMBL2029616)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383304(CHEMBL2029622)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383306(CHEMBL2029618)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383306(CHEMBL2029618)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50383313(CHEMBL2029623)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST-tagged mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed