Compile Data Set for Download or QSAR
maximum 50k data
Found 31 Enz. Inhib. hit(s) with all data for entry = 50039720
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382803(CHEMBL2023413)
Affinity DataIC50:  46nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382801(CHEMBL2023415)
Affinity DataIC50:  75nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382800(CHEMBL2023418)
Affinity DataIC50:  79nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382802(CHEMBL2023414)
Affinity DataIC50:  84nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382799(CHEMBL2023201)
Affinity DataIC50:  110nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382808(CHEMBL1933347)
Affinity DataIC50:  150nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382807(CHEMBL2023196)
Affinity DataIC50:  170nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382813(CHEMBL2023416)
Affinity DataIC50:  220nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382809(CHEMBL2023195)
Affinity DataIC50:  260nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382806(CHEMBL2023197)
Affinity DataIC50:  280nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50360581(CHEMBL1933344)
Affinity DataIC50:  390nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382805(CHEMBL2023199)
Affinity DataIC50:  400nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382804(CHEMBL2023200)
Affinity DataIC50:  410nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382810(CHEMBL2023194)
Affinity DataIC50:  970nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382814(CHEMBL2023198)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50360582(CHEMBL1933345)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382811(CHEMBL2023419)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382812(CHEMBL2023417)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of PDK1 assessed as [gamma-33P]ATP incorporation into substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382801(CHEMBL2023415)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2 using RbING as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382800(CHEMBL2023418)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2 using RbING as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382802(CHEMBL2023414)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2 using RbING as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382803(CHEMBL2023413)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2 using RbING as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382799(CHEMBL2023201)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2 using RbING as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382804(CHEMBL2023200)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2 using RbING as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382810(CHEMBL2023194)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2 using RbING as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50360582(CHEMBL1933345)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2 using RbING as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382809(CHEMBL2023195)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2 using RbING as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382808(CHEMBL1933347)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2 using RbING as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382805(CHEMBL2023199)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2 using RbING as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382806(CHEMBL2023197)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2 using RbING as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
S*Bio

Curated by ChEMBL
LigandPNGBDBM50382807(CHEMBL2023196)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2 using RbING as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed