Compile Data Set for Download or QSAR
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Found 16 Enz. Inhib. hit(s) with all data for entry = 50039951
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386758(CHEMBL2046893)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386758(CHEMBL2046893)
Affinity DataIC50:  2.51nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386755(CHEMBL2046889)
Affinity DataIC50:  15.8nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386755(CHEMBL2046889)
Affinity DataIC50:  17nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386757(CHEMBL2046892)
Affinity DataIC50:  39.8nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386757(CHEMBL2046892)
Affinity DataIC50:  44nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386756(CHEMBL2046890)
Affinity DataIC50:  62nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386756(CHEMBL2046890)
Affinity DataIC50:  63.1nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386760(CHEMBL2046895)
Affinity DataIC50:  192nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386760(CHEMBL2046895)
Affinity DataIC50:  200nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386753(CHEMBL2046891)
Affinity DataIC50:  580nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386753(CHEMBL2046891)
Affinity DataIC50:  631nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386754(CHEMBL2046888)
Affinity DataIC50:  2.79E+3nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386754(CHEMBL2046888)
Affinity DataIC50:  2.79E+3nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386759(CHEMBL2046894)
Affinity DataIC50:  7.86E+3nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50386759(CHEMBL2046894)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibition of human ERG expressed in HEK cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed