Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50039623
TargetRibosomal protein S6 kinase alpha-3(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50381078(CHEMBL2017518)
Affinity DataIC50: 252nMAssay Description:Inhibition of His-tagged RSK2 expressed in Sf9 cells using ERalpha-Ser167 RLASTND as substrate after 120 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50381083(CHEMBL2017522)
Affinity DataIC50: 356nMAssay Description:Inhibition of His-tagged RSK2 expressed in Sf9 cells using ERalpha-Ser167 RLASTND as substrate after 120 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50381082(CHEMBL2017521)
Affinity DataIC50: 493nMAssay Description:Inhibition of His-tagged RSK2 expressed in Sf9 cells using ERalpha-Ser167 RLASTND as substrate after 120 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50241294(kaempferol-3-O-(3,4-di-O-acetyl-alpha-L-rhamnopyra...)
Affinity DataIC50: 583nMAssay Description:Inhibition of His-tagged RSK2 expressed in Sf9 cells using ERalpha-Ser167 RLASTND as substrate after 120 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50381080(CHEMBL2017519)
Affinity DataIC50: 869nMAssay Description:Inhibition of His-tagged RSK2 expressed in Sf9 cells using ERalpha-Ser167 RLASTND as substrate after 120 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50381079(CHEMBL2017517)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of His-tagged RSK2 expressed in Sf9 cells using ERalpha-Ser167 RLASTND as substrate after 120 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50381084(CHEMBL2017523)
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of His-tagged RSK2 expressed in Sf9 cells using ERalpha-Ser167 RLASTND as substrate after 120 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50381081(CHEMBL2017520)
Affinity DataIC50: 1.92E+3nMAssay Description:Inhibition of His-tagged RSK2 expressed in Sf9 cells using ERalpha-Ser167 RLASTND as substrate after 120 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed