Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50039626
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381096(CHEMBL2017556)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Itk (357-620) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381092(CHEMBL2017552)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Itk (357-620) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381094(CHEMBL2017553)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Itk (357-620) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381092(CHEMBL2017552)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Syk (343 to 635) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381091(CHEMBL2017555)
Affinity DataIC50:  7nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Itk (357-620) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation coun...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381090(CHEMBL2017551)
Affinity DataIC50:  8nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Syk (343 to 635) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381097(CHEMBL2017557)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Itk (357-620) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381093(CHEMBL2017554)
Affinity DataIC50:  10.9nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Itk (357-620) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation coun...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381096(CHEMBL2017556)
Affinity DataIC50:  39.2nMAssay Description:Inhibition of Lck autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase TXK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381093(CHEMBL2017554)
Affinity DataIC50:  55.7nMAssay Description:Inhibition of Txk autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381092(CHEMBL2017552)
Affinity DataIC50:  63.9nMAssay Description:Inhibition of Lck autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase TXK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381094(CHEMBL2017553)
Affinity DataIC50:  66.5nMAssay Description:Inhibition of Txk autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase TXK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381092(CHEMBL2017552)
Affinity DataIC50:  73.8nMAssay Description:Inhibition of Txk autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase TXK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381096(CHEMBL2017556)
Affinity DataIC50:  77.5nMAssay Description:Inhibition of Txk autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381090(CHEMBL2017551)
Affinity DataIC50:  150nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Itk (357-620) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381093(CHEMBL2017554)
Affinity DataIC50:  162nMAssay Description:Inhibition of Lck autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381094(CHEMBL2017553)
Affinity DataIC50:  186nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Syk (343 to 635) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381095(CHEMBL2017550)
Affinity DataIC50:  200nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Itk (357-620) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381097(CHEMBL2017557)
Affinity DataIC50:  203nMAssay Description:Inhibition of Lck autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase TXK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381091(CHEMBL2017555)
Affinity DataIC50:  241nMAssay Description:Inhibition of Txk autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381093(CHEMBL2017554)
Affinity DataIC50:  287nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Syk (343 to 635) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381096(CHEMBL2017556)
Affinity DataIC50:  358nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Syk (343 to 635) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase TXK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381097(CHEMBL2017557)
Affinity DataIC50:  441nMAssay Description:Inhibition of Txk autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381091(CHEMBL2017555)
Affinity DataIC50:  939nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Syk (343 to 635) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381094(CHEMBL2017553)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Lck autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381097(CHEMBL2017557)
Affinity DataIC50:  2.47E+3nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Syk (343 to 635) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381091(CHEMBL2017555)
Affinity DataIC50:  3.18E+3nMAssay Description:Inhibition of Lck autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed