Compile Data Set for Download or QSAR
Report error Found 85 Enz. Inhib. hit(s) with all data for entry = 50039650
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50159165(2S,4aR,6a(R,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataEC50:  6.10nMAssay Description:Agonist activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as calcium mobilization after 1 hrs by fluorescence analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50159165(2S,4aR,6a(R,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381666(CHEMBL2022307)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as calcium mobilization after 1 hrs by fluorescence analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381677(U-69593 | CHEMBL1256748)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as calcium mobilization after 1 hrs by fluorescence analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50266337(12-epi-Salvinorin A | CHEMBL458235)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381667(CHEMBL2022018)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381666(CHEMBL2022307)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381662(CHEMBL2022302)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50266390(US8492564, 13 | CHEMBL458870 | (2S,4aR,6aR,7R,9S,1...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381656(CHEMBL2022296)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50159165(2S,4aR,6a(R,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as [35S]GTP-gamma-S binding after 3 hrs by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381668(CHEMBL2022019)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381656(CHEMBL2022296)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as calcium mobilization after 1 hrs by fluorescence analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381660(CHEMBL2022300)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381673(CHEMBL2022294)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381666(CHEMBL2022307)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as [35S]GTP-gamma-S binding after 3 hrs by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381661(CHEMBL2022301)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381657(CHEMBL2022297)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381670(CHEMBL2022021)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381665(CHEMBL2022306)
Affinity DataKi:  320nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381672(CHEMBL2022293)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381662(CHEMBL2022302)
Affinity DataEC50:  620nMAssay Description:Agonist activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as [35S]GTP-gamma-S binding after 3 hrs by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50266337(12-epi-Salvinorin A | CHEMBL458235)
Affinity DataEC50:  720nMAssay Description:Agonist activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as [35S]GTP-gamma-S binding after 3 hrs by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381656(CHEMBL2022296)
Affinity DataEC50:  730nMAssay Description:Agonist activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as [35S]GTP-gamma-S binding after 3 hrs by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381657(CHEMBL2022297)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381673(CHEMBL2022294)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381664(CHEMBL2022305)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381666(CHEMBL2022307)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381659(CHEMBL2022299)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381658(CHEMBL2022298)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381664(CHEMBL2022305)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381669(CHEMBL2022020)
Affinity DataKi:  1.07E+3nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381675(CHEMBL2022017)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381667(CHEMBL2022018)
Affinity DataEC50:  1.37E+3nMAssay Description:Agonist activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as [35S]GTP-gamma-S binding after 3 hrs by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50159165(2S,4aR,6a(R,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataKi:  1.37E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381668(CHEMBL2022019)
Affinity DataKi:  1.49E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50266390(US8492564, 13 | CHEMBL458870 | (2S,4aR,6aR,7R,9S,1...)
Affinity DataEC50:  1.63E+3nMAssay Description:Agonist activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as [35S]GTP-gamma-S binding after 3 hrs by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381665(CHEMBL2022306)
Affinity DataKi: >1.70E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381660(CHEMBL2022300)
Affinity DataEC50:  2.13E+3nMAssay Description:Agonist activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as [35S]GTP-gamma-S binding after 3 hrs by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381659(CHEMBL2022299)
Affinity DataKi:  2.26E+3nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381668(CHEMBL2022019)
Affinity DataEC50:  2.28E+3nMAssay Description:Partial agonist activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as [35S]GTP-gamma-S binding after 3 hrs by liquid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381662(CHEMBL2022302)
Affinity DataKi:  2.53E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381667(CHEMBL2022018)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381670(CHEMBL2022021)
Affinity DataKi:  3.09E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381659(CHEMBL2022299)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381672(CHEMBL2022293)
Affinity DataKi:  3.60E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381658(CHEMBL2022298)
Affinity DataKi:  4.80E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381665(CHEMBL2022306)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381674(CHEMBL2022295)
Affinity DataKi:  8.47E+3nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50381663(CHEMBL2022304)
Affinity DataKi:  9.21E+3nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
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