Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with all data for entry = 50039628
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381135(CHEMBL2017736)
Affinity DataIC50:  23nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381134(CHEMBL2017735)
Affinity DataIC50:  39nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381136(CHEMBL2017737)
Affinity DataIC50:  40nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381139(CHEMBL2017871)
Affinity DataIC50:  40nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381131(CHEMBL2017732)
Affinity DataIC50:  53nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381129(CHEMBL2017730)
Affinity DataIC50:  55nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381132(CHEMBL2017733)
Affinity DataIC50:  56nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381133(CHEMBL2017734)
Affinity DataIC50:  56nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381124(CHEMBL2017725)
Affinity DataIC50:  64nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381130(CHEMBL2017731)
Affinity DataIC50:  73nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381123(CHEMBL2017724)
Affinity DataIC50:  74nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381120(CHEMBL2017721)
Affinity DataIC50:  84nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381117(CHEMBL2017717)
Affinity DataIC50:  86nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381119(CHEMBL2017719)
Affinity DataIC50:  87nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381127(CHEMBL2017728)
Affinity DataIC50:  88nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381112(CHEMBL2017712)
Affinity DataIC50:  107nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381126(CHEMBL2017727)
Affinity DataIC50:  115nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381128(CHEMBL2017729)
Affinity DataIC50:  121nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381106(CHEMBL2017870)
Affinity DataIC50:  176nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381105(CHEMBL2017720)
Affinity DataIC50:  202nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381125(CHEMBL2017726)
Affinity DataIC50:  217nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381110(CHEMBL2017710)
Affinity DataIC50:  223nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381118(CHEMBL2017718)
Affinity DataIC50:  241nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381107(CHEMBL2017707)
Affinity DataIC50:  322nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381121(CHEMBL2017722)
Affinity DataIC50:  354nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381114(CHEMBL2017714)
Affinity DataIC50:  375nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381115(CHEMBL2017715)
Affinity DataIC50:  384nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381116(CHEMBL2017716)
Affinity DataIC50:  393nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381113(CHEMBL2017713)
Affinity DataIC50:  428nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381111(CHEMBL2017711)
Affinity DataIC50:  440nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381108(CHEMBL2017708)
Affinity DataIC50:  453nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381122(CHEMBL2017723)
Affinity DataIC50:  715nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381138(CHEMBL2017739)
Affinity DataIC50:  1.13E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381109(CHEMBL2017709)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50293701(CHEMBL549536 | N-(5-methyl-1H-pyrazol-3-yl)-2-(pyr...)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381137(CHEMBL2017738)
Affinity DataIC50:  1.99E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed