Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50039645
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381555(CHEMBL2018097)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381554(CHEMBL2018096)
Affinity DataIC50: 7.40nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381548(CHEMBL2018090)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381537(CHEMBL2017954)
Affinity DataIC50: 10nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381549(CHEMBL2018091)
Affinity DataIC50: 13nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381553(CHEMBL2018095)
Affinity DataIC50: 14nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381544(CHEMBL2018084)
Affinity DataIC50: 30nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381550(CHEMBL2018092)
Affinity DataIC50: 47nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381539(CHEMBL2017956)
Affinity DataIC50: 70nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381552(CHEMBL2018094)
Affinity DataIC50: 75nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381551(CHEMBL2018093)
Affinity DataIC50: 92nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381538(CHEMBL2017955)
Affinity DataIC50: 100nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381540(CHEMBL2018080)
Affinity DataIC50: 610nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381546(CHEMBL2018087)
Affinity DataIC50: 650nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381545(CHEMBL2018085)
Affinity DataIC50: 675nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381547(CHEMBL2018088)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381541(CHEMBL2018081)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381556(CHEMBL2018086)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381536(CHEMBL2018089)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381542(CHEMBL2018082)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50381543(CHEMBL2018083)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]AMG accumulation after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed