Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50040483
TargetLanosterol synthase(Human)
Centre Hospitalier Universitaire Vaudois (Chuv) and University of Lausanne (Unil

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50128063BDBM50128063(CHEMBL67133 | CHEMBL112210 | Allyl-{6-[3-(4-bromo-...)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of human liver microsome 2,3-OSC after 1 hr by Silica gel plate phosphor imagingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetLanosterol synthase(Human)
Centre Hospitalier Universitaire Vaudois (Chuv) and University of Lausanne (Unil

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50255431BDBM50255431(4-(trifluoromethyl)phenyl 4-(5-(allyl(methyl)amino...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human liver microsome 2,3-OSC after 1 hr by Silica gel plate phosphor imagingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetLanosterol synthase(Human)
Centre Hospitalier Universitaire Vaudois (Chuv) and University of Lausanne (Unil

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50128065BDBM50128065({4-[6-(Allyl-methyl-amino)-hexyloxy]-2-fluoro-phen...)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of human liver microsome 2,3-OSC after 1 hr by Silica gel plate phosphor imagingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetLanosterol synthase(Human)
Centre Hospitalier Universitaire Vaudois (Chuv) and University of Lausanne (Unil

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394835BDBM50394835(CHEMBL2164235)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of human liver microsome 2,3-OSC after 1 hr by Silica gel plate phosphor imagingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetLanosterol synthase(Human)
Centre Hospitalier Universitaire Vaudois (Chuv) and University of Lausanne (Unil

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50128070BDBM50128070(CHEMBL481608 | CHEMBL65230 | (4''-{[ALLYL(METHYL)A...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human liver microsome 2,3-OSC after 1 hr by Silica gel plate phosphor imagingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetLanosterol synthase(Human)
Centre Hospitalier Universitaire Vaudois (Chuv) and University of Lausanne (Unil

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394836BDBM50394836(CHEMBL2164234)
Affinity DataIC50: 10nMAssay Description:Inhibition of human liver microsome 2,3-OSC after 1 hr by Silica gel plate phosphor imagingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetLanosterol synthase(Human)
Centre Hospitalier Universitaire Vaudois (Chuv) and University of Lausanne (Unil

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394833BDBM50394833(CHEMBL2164237)
Affinity DataIC50: 11.2nMAssay Description:Inhibition of human liver microsome 2,3-OSC after 1 hr by Silica gel plate phosphor imagingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetLanosterol synthase(Human)
Centre Hospitalier Universitaire Vaudois (Chuv) and University of Lausanne (Unil

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394834BDBM50394834(CHEMBL2164236)
Affinity DataIC50: 12.7nMAssay Description:Inhibition of human liver microsome 2,3-OSC after 1 hr by Silica gel plate phosphor imagingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetLanosterol synthase(Human)
Centre Hospitalier Universitaire Vaudois (Chuv) and University of Lausanne (Unil

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50255473BDBM50255473(2-((4-(3-(4-bromophenyl)benzo[d]isothiazol-6-yloxy...)
Affinity DataIC50: 17.8nMAssay Description:Inhibition of human liver microsome 2,3-OSC after 1 hr by Silica gel plate phosphor imagingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetLanosterol synthase(Human)
Centre Hospitalier Universitaire Vaudois (Chuv) and University of Lausanne (Unil

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394832BDBM50394832(CHEMBL2164238)
Affinity DataIC50: 28.7nMAssay Description:Inhibition of human liver microsome 2,3-OSC after 1 hr by Silica gel plate phosphor imagingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed