Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50040564
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50396143(CHEMBL300739)
Affinity DataKi:  0.851nMAssay Description:Binding affinity to human recombinant 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50396145(CHEMBL300100)
Affinity DataKi:  1.26nMAssay Description:Binding affinity to human recombinant 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50396144(CHEMBL2171702)
Affinity DataKi:  9nMAssay Description:Antagonist activity at mGlu5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50396142(CHEMBL2171706)
Affinity DataKi:  13nMAssay Description:Antagonist activity at mGlu5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50396141(CHEMBL2171708)
Affinity DataKi:  20nMAssay Description:Agonist activity at GPR119More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50396140(CHEMBL2171707)
Affinity DataKi:  31nMAssay Description:Antagonist activity at mGlu5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50396139(CHEMBL2171704)
Affinity DataKi:  44nMAssay Description:Antagonist activity at mGlu5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50396138(CHEMBL2171703)
Affinity DataKi:  67nMAssay Description:Antagonist activity at mGlu5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50396137(CHEMBL2171705)
Affinity DataKi:  81nMAssay Description:Antagonist activity at mGlu5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50396136(CHEMBL2169905)
Affinity DataKi:  111nMAssay Description:Antagonist activity at mGlu5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50396146(CHEMBL51457)
Affinity DataKi:  4.37E+8nMAssay Description:Binding affinity to human recombinant 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed