Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50040147
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM14390(SILDENAFIL CITRATE | Sildenafil# | CHEMBL192 | 5-[...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389841(CHEMBL2070717)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389831(CHEMBL2070727)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389828(CHEMBL2070834)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389839(CHEMBL2070719)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM44650(1-[6-(cyanomethylsulfanyl)benzimidazolo[1,2-c]quin...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM51080(4-[(2Z)-2-(2-oxo-1-naphthalenylidene)hydrazinyl]-1...)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389837(CHEMBL2070721)
Affinity DataKi:  1.59E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389846(CHEMBL2070720)
Affinity DataKi:  1.59E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389827(CHEMBL1907082)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389832(CHEMBL2070726)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389834(CHEMBL2070725)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389845(CHEMBL1362986)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389835(CHEMBL2070724)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389830(CHEMBL1714515)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389844(CHEMBL2070728)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389829(CHEMBL2070833)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389833(CHEMBL1089322)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389836(CHEMBL2070722)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389842(CHEMBL2070723)
Affinity DataKi:  6.31E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50420172(CHEMBL2070836)
Affinity DataEC50:  2.00E+4nMAssay Description:Induction of beta-arrestin2 recruitment to human S1PR1 expressed in CHOK1 cells after 2 hrs by beta-galactosidase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389824(CHEMBL2070835)
Affinity DataKi:  2.51E+4nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50420174(CHEMBL2070837)
Affinity DataEC50:  3.16E+4nMAssay Description:Induction of beta-arrestin2 recruitment to human S1PR1 expressed in CHOK1 cells after 2 hrs by beta-galactosidase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389826(CHEMBL1620339)
Affinity DataKi:  3.98E+4nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389843(CHEMBL1622248)
Affinity DataKi:  3.98E+4nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50420173(GNF-Pf-590 | CHEMBL582739)
Affinity DataEC50:  5.01E+4nMAssay Description:Induction of beta-arrestin2 recruitment to human S1PR1 expressed in CHOK1 cells after 2 hrs by beta-galactosidase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Radboud University Nijmegen Medical Centre

Curated by ChEMBL
LigandPNGBDBM50389825(CHEMBL1626178)
Affinity DataKi:  7.94E+5nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed