Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50039857
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385224BDBM50385224(CHEMBL2037186)
Affinity DataEC50:  990nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385208BDBM50385208(CHEMBL2037327)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385207BDBM50385207(CHEMBL2037328)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385223BDBM50385223(CHEMBL2037187)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385221BDBM50385221(CHEMBL2037189)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385214BDBM50385214(CHEMBL2037313)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385201BDBM50385201(CHEMBL2037334)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385218BDBM50385218(CHEMBL2037311)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385215BDBM50385215(CHEMBL2037312)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385212BDBM50385212(CHEMBL2037315)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385213BDBM50385213(CHEMBL2037314)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385222BDBM50385222(CHEMBL2037188)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385202BDBM50385202(CHEMBL2037333)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385206BDBM50385206(CHEMBL2037329)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385210BDBM50385210(CHEMBL2037324)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385205BDBM50385205(CHEMBL2037330)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385211BDBM50385211(CHEMBL2037316)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385209BDBM50385209(CHEMBL2037325)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385219BDBM50385219(CHEMBL2037310)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385203BDBM50385203(CHEMBL2037332)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385200BDBM50385200(CHEMBL2037335)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385226BDBM50385226(CHEMBL2037326)
Affinity DataEC50:  3.40E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385220BDBM50385220(CHEMBL2037190)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385216BDBM50385216(CHEMBL2037306)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385217BDBM50385217(CHEMBL2037305)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385204BDBM50385204(CHEMBL2037331)
Affinity DataEC50:  3.90E+3nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Perugia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385225BDBM50385225(CHEMBL2037185)
Affinity DataEC50:  1.05E+4nMAssay Description:Agonist activity at human GST-tagged FXR ligand binding domain assessed as recruitment of Src-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed