TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 8.30nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 9.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 61nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 73nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 104nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: >1.40E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 1.52E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT7 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT7 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT6 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT7 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT7 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT6 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT6 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT6 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT6 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT6 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT6 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT6 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT7 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT6 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT7 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT7 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT7 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT7 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT7 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT6 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT6 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of 5HT7 receptor by radioligand displacement assayMore data for this Ligand-Target Pair