Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 50040246
TargetProtein kinase C theta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.110nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.110nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.170nMAssay Description:Inhibition of [3H]PDBu binding to PKCbeta C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.200nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.260nMAssay Description:Inhibition of [3H]PDBu binding to PKCalpha C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.380nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391388(CHEMBL2148108)
Affinity DataKi:  0.450nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391388(CHEMBL2148108)
Affinity DataKi:  0.460nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391388(CHEMBL2148108)
Affinity DataKi:  0.540nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.630nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391388(CHEMBL2148108)
Affinity DataKi:  2nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391387(CHEMBL2148107)
Affinity DataKi:  2.90nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391387(CHEMBL2148107)
Affinity DataKi:  3.30nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327946(1S,3R,5R,9R,13R)-9-Hydroxymethyl-3-[4-(3-hydroxy-p...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327946(1S,3R,5R,9R,13R)-9-Hydroxymethyl-3-[4-(3-hydroxy-p...)
Affinity DataKi:  4.40nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391388(CHEMBL2148108)
Affinity DataKi:  4.70nMAssay Description:Inhibition of [3H]PDBu binding to PKCalpha C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391388(CHEMBL2148108)
Affinity DataKi:  5.5nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391387(CHEMBL2148107)
Affinity DataKi:  5.90nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327946(1S,3R,5R,9R,13R)-9-Hydroxymethyl-3-[4-(3-hydroxy-p...)
Affinity DataKi:  7.40nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391387(CHEMBL2148107)
Affinity DataKi:  12nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391388(CHEMBL2148108)
Affinity DataKi:  12nMAssay Description:Inhibition of [3H]PDBu binding to PKCbeta C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391387(CHEMBL2148107)
Affinity DataKi:  15nMAssay Description:Inhibition of [3H]PDBu binding to PKCbeta C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391387(CHEMBL2148107)
Affinity DataKi:  15nMAssay Description:Inhibition of [3H]PDBu binding to PKCalpha C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391387(CHEMBL2148107)
Affinity DataKi:  17nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327946(1S,3R,5R,9R,13R)-9-Hydroxymethyl-3-[4-(3-hydroxy-p...)
Affinity DataKi:  25nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327946(1S,3R,5R,9R,13R)-9-Hydroxymethyl-3-[4-(3-hydroxy-p...)
Affinity DataKi:  39nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327946(1S,3R,5R,9R,13R)-9-Hydroxymethyl-3-[4-(3-hydroxy-p...)
Affinity DataKi:  63nMAssay Description:Inhibition of [3H]PDBu binding to PKCalpha C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327946(1S,3R,5R,9R,13R)-9-Hydroxymethyl-3-[4-(3-hydroxy-p...)
Affinity DataKi:  89nMAssay Description:Inhibition of [3H]PDBu binding to PKCbeta C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed