Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50039961
TargetMatrix metalloproteinase-9(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50066659(1,3-BIS-(4-METHOXY-BENZENESULFONYL)-5,5-DIMETHYL-H...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human recombinant MMP9 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386892(CHEMBL2048512 | MMP inhibitor III)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of human recombinant MMP2 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386892(CHEMBL2048512 | MMP inhibitor III)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of human recombinant MMP1 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386892(CHEMBL2048512 | MMP inhibitor III)
Affinity DataIC50: 6.40nMAssay Description:Inhibition of human recombinant MMP13 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386892(CHEMBL2048512 | MMP inhibitor III)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of human recombinant MMP12 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetStromelysin-1(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50066659(1,3-BIS-(4-METHOXY-BENZENESULFONYL)-5,5-DIMETHYL-H...)
Affinity DataIC50: 28.6nMAssay Description:Inhibition of human recombinant MMP3 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMatrix metalloproteinase-9(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50210054(3-(3,4-dihydroxy-phenyl)-acrylic acid 2-(3,4-dihyd...)
Affinity DataIC50: 610nMAssay Description:Inhibition of human recombinant MMP9 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386894(CHEMBL2048505)
Affinity DataIC50: 670nMAssay Description:Inhibition of human recombinant MMP12 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataIC50: 980nMAssay Description:Inhibition of human recombinant MMP12 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386894(CHEMBL2048505)
Affinity DataIC50: 990nMAssay Description:Inhibition of human recombinant MMP9 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386893(CHEMBL2048502)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant MMP12 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of human recombinant MMP9 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386897(CHEMBL2048508)
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of human recombinant MMP12 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386895(CHEMBL2048506)
Affinity DataIC50: 1.79E+3nMAssay Description:Inhibition of human recombinant MMP12 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50210054(3-(3,4-dihydroxy-phenyl)-acrylic acid 2-(3,4-dihyd...)
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of human recombinant MMP12 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386895(CHEMBL2048506)
Affinity DataIC50: 3.25E+3nMAssay Description:Inhibition of human recombinant MMP1 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386895(CHEMBL2048506)
Affinity DataIC50: 3.46E+3nMAssay Description:Inhibition of human recombinant MMP9 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50210054(3-(3,4-dihydroxy-phenyl)-acrylic acid 2-(3,4-dihyd...)
Affinity DataIC50: 3.58E+3nMAssay Description:Inhibition of human recombinant MMP2 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataIC50: 3.61E+3nMAssay Description:Inhibition of human recombinant MMP2 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386893(CHEMBL2048502)
Affinity DataIC50: 3.88E+3nMAssay Description:Inhibition of human recombinant MMP2 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetStromelysin-1(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 5.57E+3nMAssay Description:Inhibition of human recombinant MMP3 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataIC50: 5.62E+3nMAssay Description:Inhibition of human recombinant MMP9 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50049400((+/-)-Dihydroquercetin | 3,5,7,3',4'-pentahydroxyf...)
Affinity DataIC50: 5.75E+3nMAssay Description:Inhibition of human recombinant MMP12 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 6.68E+3nMAssay Description:Inhibition of human recombinant MMP2 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386893(CHEMBL2048502)
Affinity DataIC50: 7.62E+3nMAssay Description:Inhibition of human recombinant MMP13 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetStromelysin-1(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386894(CHEMBL2048505)
Affinity DataIC50: 8.15E+3nMAssay Description:Inhibition of human recombinant MMP3 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386896(ISOACTEOSIDE)
Affinity DataIC50: 8.22E+3nMAssay Description:Inhibition of human recombinant MMP12 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386894(CHEMBL2048505)
Affinity DataIC50: 8.23E+3nMAssay Description:Inhibition of human recombinant MMP1 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 8.46E+3nMAssay Description:Inhibition of human recombinant MMP13 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386896(ISOACTEOSIDE)
Affinity DataIC50: 8.96E+3nMAssay Description:Inhibition of human recombinant MMP2 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386897(CHEMBL2048508)
Affinity DataIC50: 9.33E+3nMAssay Description:Inhibition of human recombinant MMP13 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386902(CHEMBL2048509)
Affinity DataIC50: 9.91E+3nMAssay Description:Inhibition of human recombinant MMP9 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of human recombinant MMP13 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM76247(cid_44144307 | dihydrodaphnodorin B | [(2R,3S)-2,8...)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of human recombinant MMP9 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of human recombinant MMP12 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetStromelysin-1(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386893(CHEMBL2048502)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of human recombinant MMP3 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386898(CHEMBL2048511)
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of human recombinant MMP1 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386896(ISOACTEOSIDE)
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of human recombinant MMP13 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50155447(1,3,6,7-tetrahydroxyxantone | 1,3,6,7-Tetrahydroxy...)
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of human recombinant MMP1 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386893(CHEMBL2048502)
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of human recombinant MMP9 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386894(CHEMBL2048505)
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of human recombinant MMP2 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386897(CHEMBL2048508)
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of human recombinant MMP2 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386901(CHEMBL2048504)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of human recombinant MMP9 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386899(CHEMBL2048507)
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of human recombinant MMP13 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM76247(cid_44144307 | dihydrodaphnodorin B | [(2R,3S)-2,8...)
Affinity DataIC50: 1.41E+4nMAssay Description:Inhibition of human recombinant MMP2 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386898(CHEMBL2048511)
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of human recombinant MMP9 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386896(ISOACTEOSIDE)
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of human recombinant MMP9 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50210054(3-(3,4-dihydroxy-phenyl)-acrylic acid 2-(3,4-dihyd...)
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of human recombinant MMP1 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetStromelysin-1(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386895(CHEMBL2048506)
Affinity DataIC50: 1.48E+4nMAssay Description:Inhibition of human recombinant MMP3 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50386895(CHEMBL2048506)
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibition of human recombinant MMP2 catalytic domain incubated for 20 mins by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
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