Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50039992
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387437BDBM50387437(CHEMBL2047450)
Affinity DataKi:  5.01nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 22566BDBM22566(CHEMBL129198 | 5-chloro-2-[(4-methylpiperazin-1-yl...)
Affinity DataKi:  6.31nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387434BDBM50387434(CHEMBL2047447)
Affinity DataKi:  6.31nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133018BDBM50133018((4,5-dichloro-1H-indol-2-yl)(4-methylpiperazin-1-y...)
Affinity DataKi:  6.31nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387436BDBM50387436(CHEMBL2047449)
Affinity DataKi:  6.31nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387435BDBM50387435(CHEMBL2047448)
Affinity DataKi:  6.31nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387449BDBM50387449(CHEMBL2047466)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50132999BDBM50132999((7-Methyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)...)
Affinity DataKi:  12.6nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387438BDBM50387438(CHEMBL2047451)
Affinity DataKi:  12.6nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 26391BDBM26391(5-chloro-2-(piperazin-1-ylcarbonyl)-1H-indole | JN...)
Affinity DataKi:  12.6nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133004BDBM50133004((7-amino-1H-indol-2-yl)(4-methylpiperazin-1-yl)met...)
Affinity DataKi:  15.8nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50132996BDBM50132996((5-Fluoro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)...)
Affinity DataKi:  15.8nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387452BDBM50387452(CHEMBL2047470)
Affinity DataKi:  15.8nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387467BDBM50387467(CHEMBL2047473)
Affinity DataKi:  19.9nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387427BDBM50387427(CHEMBL2047276)
Affinity DataKi:  19.9nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133016BDBM50133016((7-Chloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)...)
Affinity DataKi:  19.9nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133020BDBM50133020((1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone |...)
Affinity DataKi:  25.1nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133007BDBM50133007((5-hydroxy-1H-indol-2-yl)(4-methylpiperazin-1-yl)m...)
Affinity DataKi:  25.1nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387424BDBM50387424(CHEMBL2047273)
Affinity DataKi:  25.1nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387469BDBM50387469(CHEMBL2047264)
Affinity DataKi:  31.6nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387459BDBM50387459(CHEMBL2047263)
Affinity DataKi:  31.6nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133001BDBM50133001((5-Amino-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-...)
Affinity DataKi:  31.6nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387451BDBM50387451(CHEMBL2047469)
Affinity DataKi:  31.6nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387464BDBM50387464(CHEMBL2047454)
Affinity DataKi:  31.6nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387446BDBM50387446(CHEMBL2047462)
Affinity DataKi:  39.8nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387471BDBM50387471(CHEMBL2047443)
Affinity DataKi:  39.8nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387440BDBM50387440(CHEMBL2047455)
Affinity DataKi:  39.8nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387455BDBM50387455(CHEMBL2047475)
Affinity DataKi:  39.8nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Mouse)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 22566BDBM22566(CHEMBL129198 | 5-chloro-2-[(4-methylpiperazin-1-yl...)
Affinity DataIC50: 40nMAssay Description:Inhibition of histamine H4 receptor-mediated chemotaxis in mouse bone marrow cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133017BDBM50133017((5-methyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)...)
Affinity DataKi:  50.1nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387450BDBM50387450(CHEMBL2047467)
Affinity DataKi:  63.1nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387475BDBM50387475(CHEMBL2047468)
Affinity DataKi:  63.1nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387426BDBM50387426(CHEMBL2047275)
Affinity DataKi:  79.4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387433BDBM50387433(CHEMBL2047446)
Affinity DataKi:  79.4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387421BDBM50387421(CHEMBL2047270)
Affinity DataKi:  79.4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387476BDBM50387476(CHEMBL2047476)
Affinity DataKi:  79.4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 22566BDBM22566(CHEMBL129198 | 5-chloro-2-[(4-methylpiperazin-1-yl...)
Affinity DataIC50: 86nMAssay Description:Inhibition of histamine H4 receptor-mediated chemotaxis in human eosinophilsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387474BDBM50387474(CHEMBL2047463)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387453BDBM50387453(CHEMBL2047471)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387461BDBM50387461(CHEMBL2047266)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387423BDBM50387423(CHEMBL2047272)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387439BDBM50387439(CHEMBL2047453)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387466BDBM50387466(CHEMBL2047259)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387472BDBM50387472(CHEMBL2047452)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387473BDBM50387473(CHEMBL2047458)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387465BDBM50387465(CHEMBL2047472)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387463BDBM50387463(CHEMBL2047268)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387441BDBM50387441(CHEMBL2047456)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387444BDBM50387444(CHEMBL2047460)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387432BDBM50387432(CHEMBL2047445)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
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