Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50040157
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50390013(CHEMBL2071529)
Affinity DataKi:  6.00E+3nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50390014(CHEMBL2071530)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM59704(1-(3,4-dichlorophenyl)-3-[4-[(3,4-dimethyl-1,2-oxa...)
Affinity DataKi:  1.30E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50390015(CHEMBL2071532)
Affinity DataKi:  2.70E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50390016(CHEMBL2071534)
Affinity DataKi:  4.20E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50390017(CHEMBL2071537)
Affinity DataKi:  4.50E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50390018(CHEMBL2071539)
Affinity DataIC50:  130nMAssay Description:Antagonist activity at human P2Y1R expressed in human 1321N1 cells assessed as inhibition of 2-MeSADP-induced increase in intracellular inositol phos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM59704(1-(3,4-dichlorophenyl)-3-[4-[(3,4-dimethyl-1,2-oxa...)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at human P2Y1R expressed in human 1321N1 cells assessed as inhibition of 2-MeSADP-induced increase in intracellular inositol phos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed