Affinity DataIC50: 63.1nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 79.4nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 79.4nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 79.4nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 79.4nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 79.4nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]ghrelin from GHS receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 398nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 631nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by IonWorks HT assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.16E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by IonWorks HT assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by IonWorks HT assayMore data for this Ligand-Target Pair