Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50040188
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390639BDBM50390639(CHEMBL2069712)
Affinity DataIC50: 331nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390640BDBM50390640(CHEMBL2069713)
Affinity DataIC50: 355nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390638BDBM50390638(CHEMBL2069711)
Affinity DataIC50: 551nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390653BDBM50390653(CHEMBL2069727)
Affinity DataIC50: 672nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390641BDBM50390641(CHEMBL2069714)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390642BDBM50390642(CHEMBL2069715)
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390645BDBM50390645(CHEMBL2069719)
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390640BDBM50390640(CHEMBL2069713)
Affinity DataIC50: 4.36E+3nMAssay Description:Inhibition of Cdk5/p25-mediated myosin heavy chain phosphorylation in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390647BDBM50390647(CHEMBL2069721)
Affinity DataIC50: 5.09E+3nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390648BDBM50390648(CHEMBL2069722)
Affinity DataIC50: 5.47E+3nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390643BDBM50390643(CHEMBL2069716)
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390654BDBM50390654(CHEMBL2069728)
Affinity DataIC50: 6.78E+3nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390655BDBM50390655(CHEMBL2069717)
Affinity DataIC50: 7.42E+3nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390651BDBM50390651(CHEMBL2069725)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390646BDBM50390646(CHEMBL2069720)
Affinity DataIC50: 8.22E+3nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390649BDBM50390649(CHEMBL2069723)
Affinity DataIC50: 8.27E+3nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390652BDBM50390652(CHEMBL2069726)
Affinity DataIC50: 8.88E+3nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390650BDBM50390650(CHEMBL2069724)
Affinity DataIC50: 9.94E+3nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Astrazeneca

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390644BDBM50390644(CHEMBL2069718)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant Cdk5/p25 incubated for 15 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed