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Found 6 Enz. Inhib. hit(s) with all data for entry = 50040254
TargetProthrombin(Bos taurus (Bovine))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50391540(CHEMBL2147469)
Affinity DataEC50:  2.10E+3nMAssay Description:Inhibition of bovine thrombin using Bz-Phe-Val-Arg-pNA as substrate incubated for 5 mins prior to substrate addition measured after 30 mins by fluori...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50391540(CHEMBL2147469)
Affinity DataEC50:  7.50E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50391541(CHEMBL2147467)
Affinity DataEC50:  700nMAssay Description:Inhibition of cathepsin B using Z-Phe-Arg-MCA as substrate incubated for 10 mins prior to substrate addition measured after 30 mins by fluorimetric a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50391540(CHEMBL2147469)
Affinity DataEC50:  4.90E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50391540(CHEMBL2147469)
Affinity DataEC50:  200nMAssay Description:Inhibition of cathepsin B using Z-Phe-Arg-MCA as substrate incubated for 10 mins prior to substrate addition measured after 30 mins by fluorimetric a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50391541(CHEMBL2147467)
Affinity DataEC50:  4.90E+3nMAssay Description:Inhibition of bovine thrombin using Bz-Phe-Val-Arg-pNA as substrate incubated for 5 mins prior to substrate addition measured after 30 mins by fluori...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed