Compile Data Set for Download or QSAR
Report error Found 174 Enz. Inhib. hit(s) with all data for entry = 50040875
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401354(CHEMBL2205805)
Affinity DataEC50:  390nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401354(CHEMBL2205805)
Affinity DataEC50:  398nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401347(CHEMBL99384)
Affinity DataEC50:  480nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401347(CHEMBL99384)
Affinity DataEC50:  501nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401348(CHEMBL593442)
Affinity DataEC50:  501nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401348(CHEMBL593442)
Affinity DataEC50:  520nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401346(CHEMBL316589 | cid_93149)
Affinity DataEC50:  631nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401352(CHEMBL2205810)
Affinity DataEC50:  631nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401352(CHEMBL2205810)
Affinity DataEC50:  670nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401346(CHEMBL316589 | cid_93149)
Affinity DataEC50:  670nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401348(CHEMBL593442)
Affinity DataEC50:  794nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401348(CHEMBL593442)
Affinity DataEC50:  850nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401347(CHEMBL99384)
Affinity DataEC50:  1.00E+3nMAssay Description:Allosteric modulation at human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401346(CHEMBL316589 | cid_93149)
Affinity DataEC50:  1.00E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401346(CHEMBL316589 | cid_93149)
Affinity DataEC50:  1.00E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401347(CHEMBL99384)
Affinity DataEC50:  1.00E+3nMAssay Description:Allosteric modulation at human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401354(CHEMBL2205805)
Affinity DataEC50:  1.20E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401352(CHEMBL2205810)
Affinity DataEC50:  1.26E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401354(CHEMBL2205805)
Affinity DataEC50:  1.26E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401352(CHEMBL2205810)
Affinity DataEC50:  1.30E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401347(CHEMBL99384)
Affinity DataEC50:  1.50E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401347(CHEMBL99384)
Affinity DataEC50:  1.58E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM64740(cid_65237 | MLS001194484 | SMR000555011 | 2,9-dime...)
Affinity DataEC50:  1.58E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM64740(cid_65237 | MLS001194484 | SMR000555011 | 2,9-dime...)
Affinity DataEC50:  1.60E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401345(CHEMBL98682)
Affinity DataEC50:  1.80E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401346(CHEMBL316589 | cid_93149)
Affinity DataEC50:  1.80E+3nMAssay Description:Allosteric modulation at human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401353(CHEMBL2205809)
Affinity DataEC50:  1.90E+3nMAssay Description:Allosteric modulation at human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401345(CHEMBL98682)
Affinity DataEC50:  2.00E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401352(CHEMBL2205810)
Affinity DataEC50:  2.00E+3nMAssay Description:Allosteric modulation at human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401344(CHEMBL317115)
Affinity DataEC50:  2.00E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401345(CHEMBL98682)
Affinity DataEC50:  2.00E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401353(CHEMBL2205809)
Affinity DataEC50:  2.00E+3nMAssay Description:Allosteric modulation at human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401346(CHEMBL316589 | cid_93149)
Affinity DataEC50:  2.00E+3nMAssay Description:Allosteric modulation at human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401344(CHEMBL317115)
Affinity DataEC50:  2.00E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401345(CHEMBL98682)
Affinity DataEC50:  2.00E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401352(CHEMBL2205810)
Affinity DataEC50:  2.20E+3nMAssay Description:Allosteric modulation at human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401351(CHEMBL2205807)
Affinity DataEC50:  2.30E+3nMAssay Description:Allosteric modulation at human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401348(CHEMBL593442)
Affinity DataEC50:  2.51E+3nMAssay Description:Allosteric modulation at human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401351(CHEMBL2205807)
Affinity DataEC50:  2.51E+3nMAssay Description:Allosteric modulation at human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401348(CHEMBL593442)
Affinity DataEC50:  2.60E+3nMAssay Description:Allosteric modulation at human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401344(CHEMBL317115)
Affinity DataEC50:  3.00E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401350(CHEMBL101165)
Affinity DataEC50:  3.16E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401344(CHEMBL317115)
Affinity DataEC50:  3.16E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401350(CHEMBL101165)
Affinity DataEC50:  3.30E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401350(CHEMBL101165)
Affinity DataEC50:  3.60E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50092158(CHEMBL415879 | cid_1318 | 1,10-phenanthroline | US...)
Affinity DataEC50:  3.90E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401350(CHEMBL101165)
Affinity DataEC50:  3.98E+3nMAssay Description:Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50092158(CHEMBL415879 | cid_1318 | 1,10-phenanthroline | US...)
Affinity DataEC50:  3.98E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401355(CHEMBL2205806)
Affinity DataEC50:  4.80E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401341(CHEMBL2205803)
Affinity DataIC50: 4.80E+3nMAssay Description:Displacement of [125I]-CCL3 from human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
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