Compile Data Set for Download or QSAR
Report error Found 74 Enz. Inhib. hit(s) with all data for entry = 50040632
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397421BDBM50397421(CHEMBL2170713)
Affinity DataEC50:  0.200nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397420BDBM50397420(CHEMBL2170563)
Affinity DataEC50:  0.600nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397419BDBM50397419(CHEMBL2170562)
Affinity DataEC50:  0.800nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50335583BDBM50335583(silvestrol | CHEMBL555196)
Affinity DataEC50:  0.800nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397418BDBM50397418(CHEMBL2170556)
Affinity DataEC50:  0.900nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397417BDBM50397417(CHEMBL2170714)
Affinity DataEC50:  1nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397416BDBM50397416(CHEMBL2170555)
Affinity DataEC50:  1nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397415BDBM50397415(CHEMBL2170703)
Affinity DataEC50:  1.20nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397414BDBM50397414(CHEMBL2170559)
Affinity DataEC50:  2nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397432BDBM50397432(CHEMBL2170560)
Affinity DataEC50:  3nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397431BDBM50397431(CHEMBL2170561)
Affinity DataEC50:  3nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397425BDBM50397425(CHEMBL2170722)
Affinity DataEC50:  3nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397413BDBM50397413(CHEMBL2170725)
Affinity DataEC50:  3nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397412BDBM50397412(CHEMBL2170718)
Affinity DataEC50:  3nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397423BDBM50397423(CHEMBL2170557)
Affinity DataEC50:  4nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397421BDBM50397421(CHEMBL2170713)
Affinity DataEC50:  4nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397436BDBM50397436(CHEMBL2170558)
Affinity DataEC50:  5nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397417BDBM50397417(CHEMBL2170714)
Affinity DataEC50:  5nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50335583BDBM50335583(silvestrol | CHEMBL555196)
Affinity DataEC50:  7nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397434BDBM50397434(AGLAFOLIN)
Affinity DataEC50:  10nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397435BDBM50397435(CHEMBL2170724)
Affinity DataEC50:  10nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397433BDBM50397433(CHEMBL2170709)
Affinity DataEC50:  11nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397413BDBM50397413(CHEMBL2170725)
Affinity DataEC50:  14nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397420BDBM50397420(CHEMBL2170563)
Affinity DataEC50:  15nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397418BDBM50397418(CHEMBL2170556)
Affinity DataEC50:  15nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397414BDBM50397414(CHEMBL2170559)
Affinity DataEC50:  17nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397432BDBM50397432(CHEMBL2170560)
Affinity DataEC50:  19nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397431BDBM50397431(CHEMBL2170561)
Affinity DataEC50:  23nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397430BDBM50397430(CHEMBL2169895)
Affinity DataEC50:  29nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397416BDBM50397416(CHEMBL2170555)
Affinity DataEC50:  30nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397429BDBM50397429(CHEMBL2170716)
Affinity DataEC50:  35nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397428BDBM50397428(CHEMBL2170719)
Affinity DataEC50:  35nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397427BDBM50397427(CHEMBL2170553)
Affinity DataEC50:  35nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397419BDBM50397419(CHEMBL2170562)
Affinity DataEC50:  35nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397415BDBM50397415(CHEMBL2170703)
Affinity DataEC50:  40nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397426BDBM50397426(CHEMBL2170708)
Affinity DataEC50:  40nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397425BDBM50397425(CHEMBL2170722)
Affinity DataEC50:  40nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397424BDBM50397424(CHEMBL2170723)
Affinity DataEC50:  50nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397412BDBM50397412(CHEMBL2170718)
Affinity DataEC50:  60nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397423BDBM50397423(CHEMBL2170557)
Affinity DataEC50:  70nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397422BDBM50397422(CHEMBL2170704)
Affinity DataEC50:  80nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397434BDBM50397434(AGLAFOLIN)
Affinity DataEC50:  90nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397436BDBM50397436(CHEMBL2170558)
Affinity DataEC50: >100nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397447BDBM50397447(CHEMBL2170717)
Affinity DataEC50:  120nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397446BDBM50397446(CHEMBL2170720)
Affinity DataEC50:  170nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397435BDBM50397435(CHEMBL2170724)
Affinity DataEC50:  200nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397445BDBM50397445(CHEMBL2170715)
Affinity DataEC50: >200nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with c-myc- 5'-UTR-luciferase construct assessed as reduction in translation initiation in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397428BDBM50397428(CHEMBL2170719)
Affinity DataEC50:  240nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397429BDBM50397429(CHEMBL2170716)
Affinity DataEC50:  275nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
Infinity Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397430BDBM50397430(CHEMBL2169895)
Affinity DataEC50:  450nMAssay Description:Inhibition of eIF4FA in human MDA-MB-231 cells transfected with tubulin 5'-UTR-luciferase construct assessed as reduction in translation initiation i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
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