Found 17 Enz. Inhib. hit(s) with all data for entry = 50040894 
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in rat brain membrane after 2.5 hrs by scintillation countingMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKi: 7.80nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in rat brain membrane after 2.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 27.5nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in rat brain membrane after 2.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in rat brain membrane after 2.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Savannah State University
Curated by ChEMBL
Savannah State University
Curated by ChEMBL
Affinity DataKi: 204nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT2B receptor after 1.5 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 249nMAssay Description:Displacement of [3H]clonidine from alpha2C adrenergic receptor after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 653nMAssay Description:Displacement of [3H]clonidine from alpha2A adrenergic receptor after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Savannah State University
Curated by ChEMBL
Savannah State University
Curated by ChEMBL
Affinity DataKi: 936nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT2B receptor after 1.5 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 945nMAssay Description:Displacement of [3H]clonidine from alpha2A adrenergic receptor after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.23E+3nMAssay Description:Displacement of [3H]clonidine from alpha2A adrenergic receptor after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.54E+3nMAssay Description:Displacement of [3H]clonidine from alpha2C adrenergic receptor after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Savannah State University
Curated by ChEMBL
Savannah State University
Curated by ChEMBL
Affinity DataKi: 2.56E+3nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5-HT2A receptor after 1.5 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Savannah State University
Curated by ChEMBL
Savannah State University
Curated by ChEMBL
Affinity DataKi: 2.77E+3nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5-HT2A receptor after 1.5 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Savannah State University
Curated by ChEMBL
Savannah State University
Curated by ChEMBL
Affinity DataKi: 2.87E+3nMAssay Description:Displacement of [3H]QNB from human recombinant M4 receptor after 1.5 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.74E+3nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D3 receptor after 1.5 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Savannah State University
Curated by ChEMBL
Savannah State University
Curated by ChEMBL
Affinity DataKi: 7.61E+3nMAssay Description:Displacement of [3H]LY278584 from human recombinant 5-HT3 receptor after 1.5 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Savannah State University
Curated by ChEMBL
Savannah State University
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]QNB from human recombinant M4 receptor after 1.5 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
