Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50040749
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399443(CHEMBL2179385)
Affinity DataIC50:  180nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399434(CHEMBL2179387)
Affinity DataIC50:  220nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399442(CHEMBL2179386)
Affinity DataIC50:  220nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399441(CHEMBL2179388)
Affinity DataIC50:  360nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399440(CHEMBL2179389)
Affinity DataIC50:  390nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399439(CHEMBL2179390)
Affinity DataIC50:  470nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399438(CHEMBL2179391)
Affinity DataIC50:  730nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399436(CHEMBL2179379)
Affinity DataIC50:  880nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399437(CHEMBL2179378)
Affinity DataIC50:  880nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399445(CHEMBL2179383)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399435(CHEMBL2179380)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399444(CHEMBL2179384)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399446(CHEMBL2179382)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399447(CHEMBL2179381)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399448(CHEMBL1230189)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399434(CHEMBL2179387)
Affinity DataKd:  4.90E+4nMAssay Description:Binding affinity to CREBBP by SPR methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed