Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50040749
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399443(CHEMBL2179385)
Affinity DataIC50: 180nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399442(CHEMBL2179386)
Affinity DataIC50: 220nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399434(CHEMBL2179387)
Affinity DataIC50: 220nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399441(CHEMBL2179388)
Affinity DataIC50: 360nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399440(CHEMBL2179389)
Affinity DataIC50: 390nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399439(CHEMBL2179390)
Affinity DataIC50: 470nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399438(CHEMBL2179391)
Affinity DataIC50: 730nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399437(CHEMBL2179378)
Affinity DataIC50: 880nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399436(CHEMBL2179379)
Affinity DataIC50: 880nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399445(CHEMBL2179383)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399435(CHEMBL2179380)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399444(CHEMBL2179384)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399446(CHEMBL2179382)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399447(CHEMBL2179381)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399448(CHEMBL1230189)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399434(CHEMBL2179387)
Affinity DataKd:  4.90E+4nMAssay Description:Binding affinity to CREBBP by SPR methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed