Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 50040963
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402953(CHEMBL2206790)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402952(CHEMBL2206791)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402951(CHEMBL2206792)
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402953(CHEMBL2206790)
Affinity DataEC50:  50.1nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402951(CHEMBL2206792)
Affinity DataEC50:  200nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402952(CHEMBL2206791)
Affinity DataEC50:  100nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402954(CHEMBL2206787)
Affinity DataEC50:  316nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402965(CHEMBL1401244)
Affinity DataEC50:  2.51E+3nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402955(CHEMBL2206785)
Affinity DataEC50:  126nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402956(CHEMBL2206784)
Affinity DataEC50:  1.58E+3nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402957(CHEMBL2206783)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402958(CHEMBL2206782)
Affinity DataEC50:  3.16E+3nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402959(CHEMBL2206781)
Affinity DataEC50:  794nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402960(CHEMBL2206780)
Affinity DataEC50:  631nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402961(CHEMBL2206779)
Affinity DataEC50:  1.58E+4nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402962(CHEMBL2206778)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402963(CHEMBL2206777)
Affinity DataEC50:  501nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402964(CHEMBL2206776)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402952(CHEMBL2206791)
Affinity DataEC50:  63.1nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402951(CHEMBL2206792)
Affinity DataEC50:  126nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402950(CHEMBL2206775)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50402953(CHEMBL2206790)
Affinity DataEC50:  100nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed