Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50042346
TargetProstaglandin E2 receptor EP1 subtype(Mouse)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424384BDBM50424384(CHEMBL2315055)
Affinity DataKd:  41nMAssay Description:Antagonist activity at mouse EP1 receptor expressed in CHOK1 cells assessed as inhibition of 17PTPGE2-induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Mouse)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424394BDBM50424394(CHEMBL1207972)
Affinity DataKd:  48nMAssay Description:Antagonist activity at mouse EP1 receptor expressed in CHOK1 cells assessed as inhibition of 17PTPGE2-induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Mouse)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424383BDBM50424383(CHEMBL2315056)
Affinity DataKd:  54nMAssay Description:Antagonist activity at mouse EP1 receptor expressed in CHOK1 cells assessed as inhibition of 17PTPGE2-induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Mouse)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424381BDBM50424381(CHEMBL2315059)
Affinity DataKd:  214nMAssay Description:Antagonist activity at mouse EP1 receptor expressed in CHOK1 cells assessed as inhibition of 17PTPGE2-induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Mouse)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424382BDBM50424382(CHEMBL2315057)
Affinity DataKd:  214nMAssay Description:Antagonist activity at mouse EP1 receptor expressed in CHOK1 cells assessed as inhibition of 17PTPGE2-induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Mouse)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424390BDBM50424390(CHEMBL2315049)
Affinity DataKd:  302nMAssay Description:Antagonist activity at mouse EP1 receptor expressed in CHOK1 cells assessed as inhibition of 17PTPGE2-induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Mouse)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424387BDBM50424387(CHEMBL2315052)
Affinity DataKd:  447nMAssay Description:Antagonist activity at mouse EP1 receptor expressed in CHOK1 cells assessed as inhibition of 17PTPGE2-induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Mouse)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424393BDBM50424393(CHEMBL2315046)
Affinity DataKd:  549nMAssay Description:Antagonist activity at mouse EP1 receptor expressed in CHOK1 cells assessed as inhibition of 17PTPGE2-induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Mouse)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424391BDBM50424391(CHEMBL2315048)
Affinity DataKd:  912nMAssay Description:Antagonist activity at mouse EP1 receptor expressed in CHOK1 cells assessed as inhibition of 17PTPGE2-induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Mouse)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424389BDBM50424389(CHEMBL2315050)
Affinity DataKd:  1.38E+3nMAssay Description:Antagonist activity at mouse EP1 receptor expressed in CHOK1 cells assessed as inhibition of 17PTPGE2-induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Mouse)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424386BDBM50424386(CHEMBL2315053)
Affinity DataKd:  2.19E+3nMAssay Description:Antagonist activity at mouse EP1 receptor expressed in CHOK1 cells assessed as inhibition of 17PTPGE2-induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Mouse)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424385BDBM50424385(CHEMBL2315054)
Affinity DataKd:  2.63E+3nMAssay Description:Antagonist activity at mouse EP1 receptor expressed in CHOK1 cells assessed as inhibition of 17PTPGE2-induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Mouse)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424388BDBM50424388(CHEMBL2315051)
Affinity DataKd:  4.36E+3nMAssay Description:Antagonist activity at mouse EP1 receptor expressed in CHOK1 cells assessed as inhibition of 17PTPGE2-induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Mouse)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424392BDBM50424392(CHEMBL2315047)
Affinity DataKd:  1.58E+4nMAssay Description:Antagonist activity at mouse EP1 receptor expressed in CHOK1 cells assessed as inhibition of 17PTPGE2-induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed